Search Result "Microtubules"


Research Article

Novel Benzo[B]Furans with Anti-Microtubule Activity Upregulate Expression of Apoptotic Genes and Arrest Leukemia Cells in G2/M Phase

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 19 Issue: 3 Year: 2019 Page: 375-388
Author(s): Karolina Królewska-Goliñska,Marcin J. Cieślak,Milena Sobczak,Rafał Dolot,Ewa Radzikowska-Cieciura,Mariola Napiórkowska,Iwona Wybrañska,Barbara Nawrot

Review Article

Targeting Tubulin-colchicine Site for Cancer Therapy: Inhibitors, Antibody- Drug Conjugates and Degradation Agents

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 1 Year: 2019 Page: 1289-1304
Author(s): Yongtao Duan,Wei Liu,Liang Tian,Yanna Mao,Chuanjun Song

Research Article

The Structure of MT189-Tubulin Complex Provides Insights into Drug Design

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 9 Year: 2019 Page: 1069-1073
Author(s): Zhongping Li,Lingling Ma,Chengyong Wu,Tao Meng,Lanping Ma,Wenyue Zheng,Yamei Yu,Qiang Chen,Jinliang Yang,Jingkang Shen

Research Article

Synthesis, Anti-proliferative Evaluation, and Molecular Docking Studies of 3-(alkylthio)-5,6-diaryl-1,2,4-triazines as Tubulin Polymerization Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 1 Year: 2019 Page: 1194-1201
Author(s): Farhad Saravani,Ebrahim Saeedian Moghadam,Hafezeh Salehabadi,Seyednasser Ostad,Morteza Pirali Hamedani,Massoud Amanlou,Mohammad Ali Faramarzi,Mohsen Amini

Novel Molecular Targets of Tauopathy; Therapeutic and Diagnostic Applications

Ebook: Frontiers in Clinical Drug Research: HIV

Volume: 8 Year: 2019
Author(s): Yasmeen M. Taalab,Mohamed El-Gamal,Mohamed Salama
Doi: 10.2174/97898114018931190801
Research Article

Expression and Interactions of Kinetoplastid Kinetochore Proteins (KKTs) from Trypanosoma brucei

Journal: Protein & Peptide Letters
Volume: 26 Issue: 1 Year: 2019 Page: 860-868
Author(s): Fangzhen Shan,Yating Diwu,Xiao Yang,Xiaoming Tu

Research Article

Impact of Hybrid-polar Histone Deacetylase Inhibitor m-Carboxycinnamic Acid bis-Hydroxyamide on Human Pancreatic Adenocarcinoma Cells

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 19 Issue: 6 Year: 2019 Page: 750-759
Author(s): Dinesh Kumar,Pranjal Sarma,Manika P. Bhadra,Anjana D. Tangutur

Review Article

Cellular Senescence-Inducing Small Molecules for Cancer Treatment

Journal: Current Cancer Drug Targets
Volume: 19 Issue: 2 Year: 2019 Page: 109-119
Author(s): Peng Liu,Yanfang Wu,Ziwen Lu,Dongsheng Shang,Zhicong Zhao,Yanting SHEN,Yafei Zhang,Feifei Zhu,Hanqing Liu,Zhigang Tu

Research Article

Differential Expression of MARK4 Protein and Related Perturbations in Females with Ovulatory PCOS

Journal: Endocrine, Metabolic & Immune Disorders - Drug Targets
Volume: 19 Issue: 7 Year: 2019 Page: 1064-1074
Author(s): Ahmad Fazilat,Nadia Rashid,Aruna Nigam,Shadab Anjum,Nimisha Gupta,Saima Wajid

Review Article

Dual Inhibitors as a New Challenge for Cancer Multidrug Resistance Treatment

Journal: Current Medicinal Chemistry
Volume: 26 Issue: 3 Year: 2019 Page: 6074-6106
Author(s): Tijana Stankovic,Jelena Dinic,Ana Podolski-Renic,Loana Musso,Sonja Stojkovic Buric,Sabrina Dallavalle,Milica Pesic

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