Search Result "MDR1"


siRNA-Mediated Knock-Down of P-Glycoprotein Expression Reveals Distinct Cellular Disposition of Anticancer Tyrosine Kinases Inhibitors

Journal: Drug Metabolism Letters
Volume: 4 Issue: 2 Year: 2010 Page: 114-119
Author(s): Amina Haouala, Holger Rumpold, Gerold Untergasser, Thierry Buclin, Hans-Beat Ris, Nicolas Widmer, Laurent A. Decosterd

Probing Multidrug Resistance P-glycoprotein Transporter Activity with SPECT Radiopharmaceuticals

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1834-1845
Author(s): David Piwnica-Worms, Vijay Sharma

Reversal of Multidrug Resistance by Natural Substances from Plants

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1757-1768
Author(s): Q. Wang, K. Michalak, O. Wesolowska, J. Deli, P. Molnar, J. Hohmann, J. Molnar, H. Engi

P-Glycoprotein, but not Multidrug Resistance Protein 4, Plays a Role in the Systemic Clearance of Irinotecan and SN-38 in Mice

Journal: Drug Metabolism Letters
Volume: 4 Issue: 4 Year: 2010 Page: 195-201
Author(s): Michael Tagen, Yanli Zhuang, Fan Zhang, K. Elaine Harstead, Jun Shen, Paula Schaiquevich, Charles H. Fraga, John C. Panetta, Christopher M. Waters, Clinton F. Stewart

Synthesis, Characterization, and Molecular Structure of a Novel Zinc (II) Complex: Assessment of Impact of MDR1Pgp Expression on its Cytotoxic Activity

Journal: Medicinal Chemistry
Volume: 6 Issue: 4 Year: 2010 Page: 191-199
Author(s): Scott E. Harpstrite, Julie L. Prior, Jothilingam Sivapackiam, Silvia D. Collins, Nigam P. Rath, Vijay Sharma

Epigenetic Regulation of ABCB1 Transporter Expression and Function

Journal: Current Pharmacogenomics and Personalized Medicine
Volume: 8 Issue: 3 Year: 2010 Page: 218-231
Author(s): Kerry Reed, Amadeo M. Parissenti

The Role of Wnt/Beta-Catenin Signaling in Renal Carcinogenesis: Lessons from Cadmium Toxicity Studies

Journal: Current Molecular Medicine
Volume: 10 Issue: 4 Year: 2010 Page: 387-404
Author(s): F. Thevenod, P.K. Chakraborty

Interplay of Metabolism and Transport in Determining Oral Drug Absorption and Gut Wall Metabolism: A Simulation Assessment Using the “Advanced Dissolution, Absorption, Metabolism (ADAM)” Model

Journal: Current Drug Metabolism
Volume: 11 Issue: 9 Year: 2010 Page: 716-729
Author(s): A. S. Darwich, S. Neuhoff, M. Jamei, A. Rostami-Hodjegan

Pharmacogenetics of Drug Transporters

Journal: Current Pharmaceutical Design
Volume: 16 Issue: 2 Year: 2010 Page: 220-230
Author(s): R. M. Franke, E. R. Gardner, A. Sparreboom

The Structure and Functions of P-Glycoprotein

Journal: Current Medicinal Chemistry
Volume: 17 Issue: 8 Year: 2010 Page: 786-800
Author(s): Y. Li, H. Yuan, K. Yang, W. Xu, W. Tang, X. Li

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