Search Result "Janus tyrosine kinase"


Multi-Kinase Inhibitors

Journal: Current Medicinal Chemistry
Volume: 22 Issue: 6 Year: 2015 Page: 695-712
Author(s): Laura Garuti,Marinella Roberti,Giovanni Bottegoni

Cancer Kinases and its Novel Inhibitors: Past, Present and Future Challenges

Journal: Current Drug Targets
Volume: 16 Issue: 11 Year: 2015 Page: 1233-1245
Author(s): Prathesha Pillai,R.S. Surenya,Shantikumar V. Nair,Vinoth-Kumar Lakshmanan

Metabolism and Disposition of Pacritinib (SB1518), an Orally Active Janus Kinase 2 Inhibitor in Preclinical Species and Humans

Journal: Drug Metabolism Letters
Volume: 9 Issue: 1 Year: 2015 Page: 28-47
Author(s): Ramesh Jayaraman,Mohammed Khalid Pasha,Anthony Williams,Kee Cee Goh,Kantharaj Ethirajulu

Review Article

Cyclin-Dependent Kinase-2 as a Target for Cancer Therapy: Progress in the Development of CDK2 Inhibitors as Anti-Cancer Agents

Journal: Current Medicinal Chemistry
Volume: 22 Issue: 2 Year: 2015 Page: 237-263
Author(s): Tahir Ali Chohan, Haiyan Qian, Youlu Pan, Jian-Zhong Chen

Hck Inhibitors as Potential Therapeutic Agents in Cancer and HIV Infection

Journal: Current Medicinal Chemistry
Volume: 22 Issue: 13 Year: 2015 Page: 1540-1564
Author(s): F. Musumeci,S. Schenone,C. Brullo,A. Desogus,L. Botta,C. Tintori

Interferon-γ-Induced Neurotoxicity of Human Astrocytes

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 14 Issue: 2 Year: 2015 Page: 251-256
Author(s): Sadayuki Hashioka,Edith G. McGeer,Tsuyoshi Miyaoka,Rei Wake,Jun Horiguchi,Patrick L. McGeer

Small Molecular Inhibitors for the Treatment of Rheumatoid Arthritis: Progress so Far

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 15 Issue: 2 Year: 2015 Page: 123-144
Author(s): Vadiraj D. Kurdekar,Hemant R. Jadhav

Endogenous Cardioprotective Agents: Role in Pre and Postconditioning

Journal: Current Drug Targets
Volume: 16 Issue: 8 Year: 2015 Page: 843-867
Author(s): Claudia Penna,Riccarda Granata,Carlo Gabriele Tocchetti,Maria Pia Gallo,Giuseppe Alloatti,Pasquale Pagliaro

Does Phosphodiesterase 11A (PDE11A) Hold Promise as a Future Therapeutic Target?

Journal: Current Pharmaceutical Design
Volume: 21 Issue: 3 Year: 2015 Page: 389-416
Author(s): Michy P. Kelly

Role of Synovial Fibroblasts in Rheumatoid Arthritis

Journal: Current Pharmaceutical Design
Volume: 21 Issue: 2 Year: 2015 Page: 130-141
Author(s): S. Lefevre,F.M.P. Meier,E. Neumann,U. Muller-Ladner

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