Search Result "Integrase"


Review Article

Recent Advances in Small-Molecule HIV-1 Integrase Inhibitors

Journal: Current Medicinal Chemistry
Volume: 28 Issue: 2 Year: 2021 Page: 4910-4934
Author(s): Chao Zhang,Qian Xie,Chi Cheong Wan,Zhe Jin,Chun Hu

Research Article

Design, Synthesis and In Vitro Evaluation of 4-Oxo-6-Substituted Phenyl- 2-Thioxo1,2,3,4-Tetrahydropyrimidine-5-Carbonitrile Derivatives as HIV Integrase Strand Transfer Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 18 Issue: 4 Year: 2021 Page: 387-395
Author(s): Pankaj Wadhwa,Priti Jain,Hemant R. Jadhav

Research Article

Novel 4-Oxo-4,10-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylic Acid Derivatives as HIV-1 Integrase Inhibitors: Synthesis, Docking Studies, Molecular Dynamics Simulation and Biological Activities

Journal: Medicinal Chemistry
Volume: 17 Issue: 9 Year: 2021 Page: 1060-1071
Author(s): Elnaz Ebrahim Zadeh,Rouhollah Vahabpour,Amirreza Dowlati Beirami,Zahra Hajimahdi,Afshin Zarghi

Review Article

A Review on Pharmacokinetics Properties of Antiretroviral Drugs toTreat HIV-1 Infections

Journal: Current Computer-Aided Drug Design
Volume: 17 Issue: 7 Year: 2021 Page: 850-864
Author(s): Sanjeev Kumar Singh,Mohd. Aqueel Khan,Krishna Kant Gupta

Research Article

Petra/Osiris/Molinspiration and Molecular Docking Analyses of 3-Hydroxy-Indolin-2-one Derivatives as Potential Antiviral Agents

Journal: Current Computer-Aided Drug Design
Volume: 17 Issue: 1 Year: 2021 Page: 123-133
Author(s): Taibi Ben Hadda,Vesna Rastija,Faisal AlMalki,Abderrahim Titi,Rachid Touzani,Yahia N. Mabkhot,Shah Khalid,Abdelkader Zarrouk,Bina S. Siddiqui

Research Article

Piroxicam Analogs: Design, Synthesis, Docking Study and Biological Evaluation as Promising Anti-HIV-1 agents

Journal: Medicinal Chemistry
Volume: 17 Issue: 0 Year: 2021 Page: 1-11
Author(s): Ali Imani,Sepehr Soleymani,Rouhollah Vahabpour,Zahra Hajimahdi,Afshin Zarghi

Research Article

Subtype Classification by Polymerase and Gag Genes of HIV-1 Iranian Sequences Registered in the NCBI GenBank

Journal: Current Proteomics
Volume: 18 Issue: 2 Year: 2021 Page: 153-161
Author(s): Behzad Dehghani,Zahra Hasanshahi,Tayebeh Hashempour,Parvin Afsar Kazerooni

Review Article

Small-molecule Inhibitors of HIV-1 Reverse Transcriptase-Associated Ribonuclease H Function: Challenges and Recent Developments

Journal: Current Medicinal Chemistry
Volume: 28 Issue: 30 Year: 2021 Page: 6146-6178
Author(s): Valentina Noemi Madia,Antonella Messore,Alessandro De Leo,Valeria Tudino,Ivano Pindinello,Francesco Saccoliti,Daniela De Vita,Luigi Scipione,Roberta Costi,Roberto Di Santo

Research Article

The Continuous Surveillance of InSTI Resistance Could be an Important Public Health Tool in the Fight Against HIV Infection

Journal: Current HIV Research
Volume: 19 Issue: 4 Year: 2021 Page: 358-367
Author(s): Giuseppa Visalli,Alessio Facciolà,Maria Giovanna Costanzo,Angela Di Pietro

Current and Promising Multiclass Drug Regimens and Long-Acting Formulation Drugs in HIV Therapy

Ebook: Foods for Special Dietary Regimens

Volume: 5 Year: 2021
Author(s): Murugesan Vanangamudi,Gnana Ruba Priya,Maida Engels
Doi: 10.2174/97898114644541200501

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