Search Result "Auto-inhibition"


Advances in peptidic and peptidomimetic-based approaches to inhibit STAT signaling in human diseases

Journal: Current Protein & Peptide Science
Volume: 17 Issue: 2 Year: 2016 Page: 135-146
Author(s): Malgorzata Szelag,Joanna Wesoly,Hans A.R. Bluyssen

open access plus

Identification of Protein Palmitoylation Inhibitors from a Scaffold Ranking Library

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 19 Issue: 4 Year: 2016 Page: 262-274
Author(s): Laura D. Hamel,Brian J. Lenhart,David A. Mitchell,Radleigh G. Santos,Marc A. Giulianotti,Robert J. Deschenes

Escape, or Vanish: Control the Fate of p53 through MDM2-Mediated Ubiquitination

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2016 Page: 174-189
Author(s): Jinlian Wei,Yingrui Yang,Mengchen Lu,Lili Xu,Fang Liu,Zhenwei Yuan,Qichao Bao,Zhengyu Jiang,Xiaoli Xu,Xiaoke Guo,Xiaojin Zhang,Qidong You,Haopeng Sun

Review Article

Structural Insights into IRE1 Functions in the Unfolded Protein Response

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 41 Year: 2016 Page: 4706-4716
Author(s): Jianqiong Yang,Haiqing Liu,Linfu Li,Hai Liu,Weimei Shi,Xiaoliang Yuan,Longhuo Wu

Protein Knockdown Technology: Application of Ubiquitin Ligase to Cancer Therapy

Journal: Current Cancer Drug Targets
Volume: 16 Issue: 2 Year: 2016 Page: 136-146
Author(s): Nobumichi Ohoka,Norihito Shibata,Takayuki Hattori,Mikihiko Naito

Review Article

Traumatic Brain Injury and Blood-Brain Barrier Cross-Talk

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 15 Issue: 9 Year: 2016 Page: 1030-1044
Author(s): Mohammad Nasser, Fabienne Bejjani, Mohamad Raad, Hadi Abou-El-Hassan, Sarah Mantash, Amaly Nokkari, Naify Ramadan, Nouhad Kassem, Stefania Mondello, Eva Hamade, Hala Darwish, Kazem Zibara, Firas Kobeissy

Drugs Targeting the Canonical NF-κB Pathway to Treat Viral and Autoimmune Myocarditis

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 4 Year: 2016 Page: 440-449
Author(s): Alan Valaperti

Acute Lymphoblastic Leukemia and Regulatory T cells: Biomarkers and Immunopathogenesis

Journal: Current Immunology Reviews (Discontinued)
Volume: 12 Issue: 1 Year: 2016 Page: 14-19
Author(s): Carlos H. Hiroki,Rafaela P. Erthal,Ana P.L. Pereira,Letícia M. Pacholak,Thiago C. Fujita,Poliana C. Marinello,Idessânia N. Costa,Sérgio P.D. da Rocha,Maria A.E. Watanabe,Carlos E.C. de Oliveira

Enzyme Activity Assays for Protein Kinases: Strategies to Identify Active Substrates

Journal: Current Drug Discovery Technologies
Volume: 13 Issue: 1 Year: 2016 Page: 2-15
Author(s): Brad A. Haubrich,David C. Swinney

Good at Heart: Preserving Cardiac Metabolism during aging

Journal: Current Diabetes Reviews
Volume: 12 Issue: 2 Year: 2016 Page: 90-99
Author(s): Daniela Sorriento,Antonietta Franco,Maria Rosaria Rusciano,Angela Serena Maione,Maria Soprano,Maddalena Illario,Guido Iaccarino,Michele Ciccarelli

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