Search Result "Acetylcholinesterase inhibition"


TRISOXIME – a Bulky Trisquaternary Reactivator of Acetylcholinesterase

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 5 Year: 2016 Page: 372-375
Author(s): Kamil Kuca,Kamil Musilek,Daniel Jun

Research Article

Inhibition of Aβ(1-42)Oligomerization, Fibrillization and Acetylcholinesterase Activity by Some Anti-Inflammatory Drugs: An in vitro Study

Journal: Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry
Volume: 15 Issue: 3 Year: 2016 Page: 191-203
Author(s): Hamendra S. Parmar,Anshul Assaiya,Renuka Agrawal,Shalini Tiwari,Iram Mufti,Neha Jain,Elangovan Manivannan,Tushar Banerjee,Anil Kumar

Monooxime Bispyridinium Reactivators Bearing Xylene Linker Synthesis and In Vitro Evaluation on Model of Organophosphate-Inhibited Acetylcholinesterase

Journal: Medicinal Chemistry
Volume: 12 Issue: 4 Year: 2016 Page: 362-370
Author(s): Kamil Musilek,Jan Hambalek,Ondrej Holas,Vlastimil Dohnal,Kamil Kuca

Flexibility in the Molecular Design of Acetylcholinesterase Reactivators: Probing Representative Conformations by Chemometric Techniques and Docking/QM Calculations

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 5 Year: 2016 Page: 360-371
Author(s): Willian E.A. de Lima,Ander F. Pereira,Alexandre A. de Castro,Elaine F.F. da Cunha,Teodorico C. Ramalho

AChE Inhibition-based Multi-target-directed Ligands, a Novel Pharmacological Approach for the Symptomatic and Disease-modifying Therapy of Alzheimer’s Disease

Journal: Current Neuropharmacology
Volume: 14 Issue: 4 Year: 2016 Page: 364-375
Author(s): Yu Wang,Hao Wang,Hong-zhuan Chen

Chemical Composition and Inhibitory Effects of Hypericum brasiliense and H. connatum on Prolyl Oligopeptidase and Acetylcholinesterase Activities

Journal: Medicinal Chemistry
Volume: 12 Issue: 5 Year: 2016 Page: 457-463
Author(s): Maura Z. dos Santos,Ionara I. Dalcol,Luciana Adolpho,Meritxell Teixidó,Teresa Tarragó,Ademir Morel,Ernest Giralt

Research Article

An Investigation of Sodium Fusidate and Recombinant Cytochrome P450 Enzymes Inhibition In-Vitro

Journal: Drug Metabolism Letters
Volume: 10 Issue: 3 Year: 2016 Page: 180-186
Author(s): John Mishriky, Jacqueline Balassone, Zenah Bashour, Simranjit Kaur, Vini Raman, Robel Getachew, Narin Osman, Daniel Guidone, Vincent Chan, Peter J. Little

Research Article

In Silico Analysis of Green Tea Polyphenols as Inhibitors of AChE and BChE Enzymes in Alzheimer’s Disease Treatment

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 15 Issue: 5 Year: 2016 Page: 624-628
Author(s): Babar Ali,Qazi M.S. Jamal,Saiba Shams,Naser A. Al-Wabel,Mughees U. Siddiqui,Mohammad A. Alzohairy,Mohammed A. Al Karaawi,Kavindra Kumar Kesari,Gohar Mushtaq,Mohammad A. Kamal

Biological Evaluation of Azomethine-dihydroquinazolinone Conjugates as Cancer and Cholinesterase Inhibitors

Journal: Medicinal Chemistry
Volume: 12 Issue: 1 Year: 2016 Page: 74-82
Author(s): Jamshed Iqbal,Aamer Saeed,Syed J.A. Shah,Mariya al-Rashida,Shams-ul Mahmood

Withanolides: Biologically Active Constituents in the Treatment of Alzheimer’s Disease

Journal: Medicinal Chemistry
Volume: 12 Issue: 3 Year: 2016 Page: 238-256
Author(s): Shahid A. Khan,Sher B. Khan,Zarbad Shah,Abdullah M. Asiri

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