Search Result "3-triazoles"


Research Article

Design, Synthesis and in silico Studies of New 5-substituted-2-(2-(5-aryl- 1H-1, 2, 4-triazole-3-ylthio) acetyl) Hydrazine Carbothioamide/ Carboxamides for Anticonvulsant Activity

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 10 Year: 2017 Page: 1155-1163
Author(s): Radhika Chelamalla,Ajitha Makula,Sarangapani Manda

Research Article

1,2,3-Triazole-Isoxazole Based Acetylcholinesterase Inhibitors: Synthesis, Biological Evaluation and Docking Study

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 58-65
Author(s): Zahra Najafi,Mohammad Mahdavi,Mina Saeedi,Reyhaneh Sabourian,Mahnaz Khanavi,Maliheh Safavi,Maliheh Barazandeh Tehrani,Abbas Shafiee,Alireza Foroumadi,Tahmineh Akbarzadeh

Research Article

Possible Binding Mode Analysis of Pyrazolo-triazole Hybrids as Potential Anticancer Agents through Validated Molecular Docking and 3D-QSAR Modeling Approaches

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 5 Year: 2017 Page: 515-527
Author(s): Siekh Abdul Amin,Nilanjan Adhikari,Ram K. Agrawal,Tarun Jha,Shovanlal Gayen

Research Article

In vitro α-Glucosidase Inhibition by Non-sugar based Triazoles of Dibenzoazepine, their Structure-Activity Relationship, and Molecular Docking

Journal: Medicinal Chemistry
Volume: 13 Issue: 7 Year: 2017 Page: 698-704
Author(s): Maria A. Khan,Kulsoom Javaid,Abdul Wadood,Alam Jamal,Farhana Batool,Saba Fazal-ur-Rehman,Fatima Z. Basha,Muhammad I. Choudhary

Research Article

Synthesis and Biological Evaluation of Triazole-Vanillin Molecular Hybrids as Anti-Cancer Agents

Journal: Current Bioactive Compounds
Volume: 13 Issue: 3 Year: 2017 Page: 223-235
Author(s): Gangavaram V. M. Sharma,Kandikonda S. Kumar,Sheri V. Reddy,Arumugam Nagalingam,Kathleen M. Cunningham,Ramesh Ummanni,Helmut Hugel,Dipali Sharma,Sanjay V. Malhotra

Research Article

Synthesis, Antibacterial, Antifungal, Antimycobacterial Activity Evaluation of Novel 1,2,4-triazole Derivatives Bearing 4-Aminophenyl Moiety

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 8 Year: 2017 Page: 938-948
Author(s): Betul Kaya Cavusoglu,Leyla Yurttas,Meral Y. Cankilic,Zafer A. Kaplancikli

Research Article

Discovery of Flexible Naphthyltriazolylmethane-based Thioacetic Acids as Highly Active Uric Acid Transporter 1 (URAT1) Inhibitors for the Treatment of Hyperuricemia of Gout

Journal: Medicinal Chemistry
Volume: 13 Issue: 3 Year: 2017 Page: 260-281
Author(s): Xiansheng Zhang,Jingwei Wu,Wei Liu,Yuqiang Liu,Yafei Xie,Qian Shang,Zhixing Zhou,Weiren Xu,Lida Tang,Jianwu Wang,Guilong Zhao

Research Article

Synthesis of New Symmetrical N, N'-Diacylhydrazines and 2-(1,2,3- Triazol-4-yl)-1,3,4-oxadiazoles

Journal: Letters in Organic Chemistry
Volume: 14 Issue: 8 Year: 2017 Page: 591-596
Author(s): Bakr F. Abdel-Wahab,Mohammad Hayal Alotaibi,Gamal A. El-Hiti

Review Article

Recent Advances in Synthesis and Biological Activity of Modified Cap Analogs

Journal: Current Organic Chemistry
Volume: 21 Issue: 25 Year: 2017 Page: 2530-2560
Author(s): Muthian Shanmugasundaram,Annamalai Senthilvelan,Anilkumar R. Kore

Research Article

New Cyclopenta[4,5]pyrido[3,2:4,5]thieno[2,3-e][1,2,4]triazolo[4,3-c]pyrimidines and Cyclopenta[4,5]pyrido[3,2:4,5]thieno[2,3-e][1,2,4]triazolo[1,5-c]pyrimidines: Synthesis and Antimicrobial Activities

Journal: Current Organic Chemistry
Volume: 21 Issue: 1 Year: 2017 Page: 1227-1241
Author(s): Samvel N. Sirakanyan,Domenico Spinelli,Athina Geronikaki,Viktor A. Kartsev,Elmira K. Hakobyan,Henrik A. Panosyan,Hrachya M. Stepanyan,Luca Zuppiroli,Anush A. Hovakimyan

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