Search Result "3]triazole-4"


Research Article

Design, Synthesis and in silico Studies of New 5-substituted-2-(2-(5-aryl- 1H-1, 2, 4-triazole-3-ylthio) acetyl) Hydrazine Carbothioamide/ Carboxamides for Anticonvulsant Activity

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 10 Year: 2017 Page: 1155-1163
Author(s): Radhika Chelamalla,Ajitha Makula,Sarangapani Manda

Research Article

1,2,3-Triazole-Isoxazole Based Acetylcholinesterase Inhibitors: Synthesis, Biological Evaluation and Docking Study

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 58-65
Author(s): Zahra Najafi,Mohammad Mahdavi,Mina Saeedi,Reyhaneh Sabourian,Mahnaz Khanavi,Maliheh Safavi,Maliheh Barazandeh Tehrani,Abbas Shafiee,Alireza Foroumadi,Tahmineh Akbarzadeh

Research Article

Synthesis, Antibacterial, Antifungal, Antimycobacterial Activity Evaluation of Novel 1,2,4-triazole Derivatives Bearing 4-Aminophenyl Moiety

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 8 Year: 2017 Page: 938-948
Author(s): Betul Kaya Cavusoglu,Leyla Yurttas,Meral Y. Cankilic,Zafer A. Kaplancikli

Research Article

Possible Binding Mode Analysis of Pyrazolo-triazole Hybrids as Potential Anticancer Agents through Validated Molecular Docking and 3D-QSAR Modeling Approaches

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 5 Year: 2017 Page: 515-527
Author(s): Siekh Abdul Amin,Nilanjan Adhikari,Ram K. Agrawal,Tarun Jha,Shovanlal Gayen

Research Article

Discovery of Flexible Naphthyltriazolylmethane-based Thioacetic Acids as Highly Active Uric Acid Transporter 1 (URAT1) Inhibitors for the Treatment of Hyperuricemia of Gout

Journal: Medicinal Chemistry
Volume: 13 Issue: 3 Year: 2017 Page: 260-281
Author(s): Xiansheng Zhang,Jingwei Wu,Wei Liu,Yuqiang Liu,Yafei Xie,Qian Shang,Zhixing Zhou,Weiren Xu,Lida Tang,Jianwu Wang,Guilong Zhao

Research Article

Synthesis of New Symmetrical N, N'-Diacylhydrazines and 2-(1,2,3- Triazol-4-yl)-1,3,4-oxadiazoles

Journal: Letters in Organic Chemistry
Volume: 14 Issue: 8 Year: 2017 Page: 591-596
Author(s): Bakr F. Abdel-Wahab,Mohammad Hayal Alotaibi,Gamal A. El-Hiti

Research Article

New Cyclopenta[4,5]pyrido[3,2:4,5]thieno[2,3-e][1,2,4]triazolo[4,3-c]pyrimidines and Cyclopenta[4,5]pyrido[3,2:4,5]thieno[2,3-e][1,2,4]triazolo[1,5-c]pyrimidines: Synthesis and Antimicrobial Activities

Journal: Current Organic Chemistry
Volume: 21 Issue: 1 Year: 2017 Page: 1227-1241
Author(s): Samvel N. Sirakanyan,Domenico Spinelli,Athina Geronikaki,Viktor A. Kartsev,Elmira K. Hakobyan,Henrik A. Panosyan,Hrachya M. Stepanyan,Luca Zuppiroli,Anush A. Hovakimyan

Research Article

Synthesis and Evaluation of A New Series of Thiazole Derivatives as Potential Antitumor Agents and MMP Inhibitors

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 5 Year: 2017 Page: 674-681
Author(s): Zafer Asim Kaplancikli,Mehlika Dilek Altıntop,Ozlem Atli,Belgin Sever,Merve Baysal,Halide Edip Temel,Fatih Demirci,Ahmet Ozdemir

Research Article

Novel [1,2,4] Triazol [4,3-a] Pyridine Derivatives as Potential Selective c-Met Inhibitors with Improved Pharmacokinetic Properties

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 8 Year: 2017 Page: 1102-1112
Author(s): Junjun Zhao,Shaohua Gou,Xiaobing Zhang,Yan Liang,Lei Fang

Research Article

The Oxime Derivatives of 1-R-1H-Naphtho[2,3-d][1,2,3]triazole-4,9-dione 2-oxides: Synthesis and Properties

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 1 Year: 2017 Page: 1814-1823
Author(s): Leonid M. Gornostaev,Vladimir B. Tsvetkov,Alina A. Markova,Tatyana I. Lavrikova,Yulia G. Khalyavina,Anastasia S. Kuznetsova,Dmitry N. Kaluzhny,Alexei V. Shunayev,Maria V. Tsvetkova,Valeria A. Glazunova,Vladimir V. Chernyshev,Alexander A. Shtil

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