Search Result "saquinavir"


Comparative Efflux of Saquinavir, Ritonavir and Lopinavir from Primary Human Cells

Journal: Drug Metabolism Letters
Volume: 4 Issue: 4 Year: 2010 Page: 241-245
Author(s): Bilge Diker, Omar Janneh, Rolf P.G. van Heeswijk, Karen F.T. Copeland

Enhancing the Delivery of Anti Retroviral Drug “Saquinavir” Across the Blood Brain Barrier Using Nanoparticles

Journal: Current HIV Research
Volume: 8 Issue: 5 Year: 2010 Page: 396-404
Author(s): Supriya D. Mahajan, Indrajit Roy, GaiXia Xu, Ken-Tye Yong, Hong Ding, Ravikumar Aalinkeel, Jessica L. Reynolds, Donald E. Sykes, Bindukumar B. Nair, Elaine Y. Lin, Paras N. Prasad, Stanley A. Schwartz

Research Article

CoMFA, CoMSIA and Docking Studies of Saquinavir Based Peptidomimetic Inhibitors of HIV-1 Protease

Journal: Current Enzyme Inhibition
Volume: 12 Issue: 2 Year: 2016 Page: 161-169
Author(s): Vandana Saini, Sakshi Piplani, Amita S. Dang, Ajit Kumar

Saquinavir/Ritonavir Monotherapy as a New Nucleoside-Sparing Maintenance Strategy in Long-Term Virologically Suppressed HIVInfected Patients

Journal: Current HIV Research
Volume: 8 Issue: 6 Year: 2010 Page: 467-470
Author(s): Patricia Echeverria, Pere Domingo, Mar Gutierrez, Mateo Gracia, Monse Fuster, Jose Molto, Jordi Puig, Nuria Perez-Alvarez, Bonaventura Clotet, Eugenia Negredo

Research Article

Molecular Docking, DFT Studies and ADMET Simulations for Evaluating Already Approved FDA Drugs as Inhibitors for SARS-Cov-2 RNADependent Polymerase

Journal: Letters in Drug Design & Discovery
Volume: 18 Issue: 7 Year: 2021 Page: 674-685
Author(s): Manos C. Vlasiou,Kyriakos I. Ioannou,Kyriaki S. Pafiti

The Secreted Aspartic Proteinases as a New Target in the Therapy of Candidiasis

Journal: Current Drug Targets
Volume: 3 Issue: 5 Year: 2002 Page: 351-357
Author(s): M. Bein, M. Schaller, H.C. Korting

Successful Applications of Computer Aided Drug Discovery: Moving Drugs from Concept to the Clinic

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 127-141
Author(s): Tanaji T. Talele, Santosh A. Khedkar, Alan C. Rigby

Inhibitors of HIV-1 Protease: Current State of the Art 10 Years After their Introduction. From Antiretroviral Drugs to Antifungal, Antibacterial and Antitumor Agents Based on Aspartic Protease Inhibitors

Journal: Current Medicinal Chemistry
Volume: 14 Issue: 2 Year: 2007 Page: 2734-2748
Author(s): Antonio Mastrolorenzo, Stefano Rusconi, Andrea Scozzafava, Giuseppe Barbaro, Claudiu T. Supuran

Nucleoside-Free Boosted Double PI Regimen: Significant CD4+ T-Cell Recovery in Patients with Poor Immunologic Response Despite Virologic Suppression

Journal: Current HIV Research
Volume: 6 Issue: 6 Year: 2008 Page: 555-559
Author(s): Clara Lehmann, Norma Jung, Anika Hofmann, Oliver A. Cornely, Christoph Wyen, Gerd Fatkenheuer, Pia Hartmann

Current Development on HIV-1 Protease Inhibitors

Journal: Current Computer-Aided Drug Design
Volume: 3 Issue: 3 Year: 2007 Page: 201-213
Author(s): Ornjira Aruksakunwong, Siriporn Promsri, Kitiyaporn Wittayanarakul, Piyarat Nimmanpipug, Vannajan S. Lee, Atchara Wijitkosoom, Pornthep Sompornpisut, Supot Hannongbua

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