Search Result "roscovitine"


Cyclin-dependent kinase Inhibitors Inspired by Roscovitine: Purine Bioisosteres

Journal: Current Pharmaceutical Design
Volume: 18 Issue: 20 Year: 2012 Page: 2974-2980
Author(s): Radek Jorda,Kamil Paruch,Vladimir Krystof

CDK Inhibitors Induce Mitochondria-mediated Apoptosis Through the Activation of Polyamine Catabolic Pathway in LNCaP, DU145 and PC3 Prostate Cancer Cells

Journal: Current Pharmaceutical Design
Volume: 20 Issue: 2 Year: 2014 Page: 180-188
Author(s): Elif Damla Arisan, Pinar Obakan, Ajda Coker-Gurkan, Annarica Calcabrini, Enzo Agostinelli, Narcin Palavan Unsal

Research Article

Novel Pyrazolo[3,4-d]pyrimidines as Potential Cytotoxic Agents: Design, Synthesis, Molecular Docking and CDK2 Inhibition

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 19 Issue: 1 Year: 2019 Page: 1368-1381
Author(s): Mai Maher,Asmaa E. Kassab,Ashraf F. Zaher,Zeinab Mahmoud

Structural Basis for Interaction of Inhibitors with Cyclin-Dependent Kinase 2

Journal: Current Computer-Aided Drug Design
Volume: 1 Issue: 1 Year: 2005 Page: 53-64
Author(s): Fernanda Canduri, Walter Filgueira de Azevedo Jr.

Pharmacological Cyclin-Dependent Kinase Inhibitors (PCIs) as Potential Antiviral Drugs

Journal: Anti-Infective Agents in Medicinal Chemistry
Volume: 5 Issue: 4 Year: 2006 Page: 345-355
Author(s): L. M. Schang

Research Article

Novel Therapeutic Approach in Acute Promyelocytic Leukemia with All-trans retinoic Acid and Cyclin-dependent Kinase Inhibitors

Journal: Clinical Cancer Drugs
Volume: 5 Issue: 1 Year: 2018 Page: 50-59
Author(s): G. Tsolkas,D. Komninou,E. Briasoulis,E. Hatzimichael,N.A. Papanikolaou

Cyclin-Dependent Kinase Inhibitors as Anticancer Drugs

Journal: Current Drug Targets
Volume: 11 Issue: 3 Year: 2010 Page: 291-302
Author(s): Vladimir Krystof, Stjepan Uldrijan

Inhibitors of Cyclin-Dependent Kinases: Potential Drugs for the Treatment of Neurodegenerative Disorders?

Journal: Current Medicinal Chemistry - Central Nervous System Agents
Volume: 5 Issue: 2 Year: 2005 Page: 101-109
Author(s): Merce Pallas, Anna M. Canudas, Ester Verdaguer, Clemens Allgaier, Susana Garcia de Arriba, Daniel Alvira, Francesc X. Sureda, Antoni Camins

Drugging Cell Cycle Kinases in Cancer Therapy

Journal: Current Drug Targets
Volume: 6 Issue: 3 Year: 2005 Page: 325-335
Author(s): S. Blagden, J. de Bono

Role of the HIV-1 Positive Elongation Factor P-TEFb and Inhibitors Thereof

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 9 Issue: 3 Year: 2009 Page: 379-385
Author(s): Yan Wang, Xin-yong Liu, Erik De Clercq

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