Search Result "falcipains"


Falcipain Inhibition as a Promising Antimalarial Target

Journal: Current Topics in Medicinal Chemistry
Volume: 12 Issue: 5 Year: 2012 Page: 408-444
Author(s): Maria Marco, Jose Miguel Coteron

Mini-Review Article

Falcipain-2 and Falcipain-3 Inhibitors as Promising Antimalarial Agents

Journal: Current Medicinal Chemistry
Volume: 28 Issue: 1 Year: 2021 Page: 3037-3058
Author(s): Roberta Ettari,Santo Previti,Carla Di Chio,Maria Zappalà

Falcipains, Plasmodium falciparum Cysteine Proteases as Key Drug Targets Against Malaria

Journal: Current Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2011 Page: 1555-1572
Author(s): C. Teixeira, J. R.B. Gomes, P. Gomes

Design, Synthesis and Preliminary Screening of Some New Conformationally Constrained Falcipain-2 Inhibitors as Potential Antimalarial Agents

Journal: Letters in Drug Design & Discovery
Volume: 6 Issue: 4 Year: 2009 Page: 258-267
Author(s): Anil K. Shinde, Bishram S. Chouhan, Shirshendu Dasgupta, Rajani Giridhar, Philip Rosenthal, Jiri Gut, Mange R. Yadav

Profiling the Structural Determinants of Heteroarylnitrile Scaffold-Based Derivatives as Falcipain-2 Inhibitors by In Silico Methods

Journal: Current Medicinal Chemistry
Volume: 20 Issue: 1 Year: 2013 Page: 2032-2042
Author(s): Jinghui Wang, Yan Li, Yinfeng Yang, Shuwei Zhang, Ling Yang

Research Article

Combined CADD and Virtual Screening to Identify Novel Nonpeptidic Falcipain-2 Inhibitors

Journal: Current Computer-Aided Drug Design
Volume: 17 Issue: 4 Year: 2021 Page: 579-588
Author(s): Trisha Rajguru,Dipshikha Bora,Mahendra Kumar Modi

Oxidation and Tyrosine Nitration Induce Structural Changes and Inhibits Plasmodium falciparum Falcipain-2 Activity In Vitro

Journal: Protein & Peptide Letters
Volume: 23 Issue: 6 Year: 2016 Page: 562-572
Author(s): Jean B. Bertoldo,Hernán Terenzi

Review Article

Targeting Cysteine Proteases from Plasmodium falciparum: A General Overview, Rational Drug Design and Computational Approaches for Drug Discovery

Journal: Current Drug Targets
Volume: 19 Issue: 5 Year: 2018 Page: 501-526
Author(s): Boris D. Bekono,Fidele Ntie-Kang,Luc C. Owono Owono,Eugene Megnassan

Research Article

Inhibition of Hemoglobin Degrading Protease Falcipain-2 as a Mechanism for Anti-Malarial Activity of Triazole-Amino Acid Hybrids

Journal: Current Topics in Medicinal Chemistry
Volume: 20 Issue: 5 Year: 2020 Page: 377-389
Author(s): Vigyasa Singh,Rahul Singh Hada,Amad Uddin,Babita Aneja,Mohammad Abid,Kailash C. Pande,Shailja Singh

Cysteine Proteases of Malaria Parasites: Targets for Chemotherapy

Journal: Current Pharmaceutical Design
Volume: 8 Issue: 1 Year: 2002 Page: 1659-1672
Author(s): Philip J. Rosenthal, Puran S. Sijwali, Ajay Singh, Bhaskar R. Shenai

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