Anti-Infective Agents

Anti-Infective Agents in Medicinal Chemistry

Editor-in-Chief:

Giovanni Gherardi
University Bio-Medico
Rome
Italy

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Open Access Articles

Development of Usnic Acid Embedded Eudragit Microspheres for Alleviation of Nosocomial Infections open Access plus

Volume: 18   Issue: 1
Pp: 79-87
Shraddha Pandey*, Shashi K. Misra and Nisha Sharma
DOI:10.2174/2211352517666190126161205

Synergistic Effects of Essential Oils of Ammoides verticillata and Satureja candidissima Against Many Pathogenic Microorganisms open Access plus

Volume: 18   Issue: 1
Pp: 72-78
Fatima Benyoucef, Mohammed El Amine Dib*, Boufeldja Tabti, Arrar Zoheir, Jean Costa and Alain Muselli
DOI:10.2174/2211352517666190227161811

Solid State Kinetics, Spectroscopic, Thermal Degradation and Fungicidal Studies of Biodegradable Copper Surfactants Derived from Lauric Acid open Access plus

Volume: 18   Issue: 1
Pp: 59-71
Shilpa Jain, Rashmi Sharma and Arun K. Sharma*
DOI:10.2174/2211352517666190514074750

Immunostimulating Activity of Gold-modified Nanodiamond Particles open Access plus

Volume: 18   Issue: 1
Pp: 54-58
Evgenii Plotnikov*, Skoryk Nina, Savelyev Daniil and Vladimir Plotnikov
DOI:10.2174/2211352517666190328122008

Effect of Chitosan, Chitosan Nanoparticle, Anacyclus pyrethrum and Cyperus rotundus in Combating Plasmid Mediated Resistance in Periodontitis open Access plus

Volume: 18   Issue: 1
Pp: 43-53
Usha Subbiah*, Gokulalakshmi Elayaperumal, Sonaa Elango, Arvind Ramanathan, Bagavad Gita and Karthikeyan Subramani
DOI:10.2174/2211352517666190221150743

Design, Optimization, Synthesis and AntiTB Screening of Benzimidazole Derivatives open Access plus

Volume: 18   Issue: 1
Pp: 24-42
Theivendren Panneerselvam, Selvaraj Kunjiappan, Veerachamy Alagarsamy, Govindaraj Saravanan* and Pavadai Parasuraman
DOI:10.2174/2211352517666190301144054

Punica granatum L. (Pomegranate): A Potential Anti-microbial Agent open Access plus

Volume: 18   Issue: 1
Pp: 2-14
Aida Doostkam, Kamyar Iravani and Shahindokht Bassiri-Jahromi*
DOI:10.2174/2211352517666190215113232

Synthesis, In-Vitro and In-Silico Studies of Benzothiazole Azo-Ester Derivatives as Anti-TB Agents open Access plus

Volume: 18   Issue: 1
Pp: 15-23
Mahesh Bhat* and Shiddappa L. Belagali
DOI:10.2174/2211352517666190126160534

Deboronation of New Clarithromycin-Benzo[c][1,2]oxaborole Conjugates open Access plus

Volume: 17   Issue: 2
Pp: 99-104
Gennady B. Lapa*, Elena B. Isakova, Elena B. Mirchink and Maria N. Preobrazhenskaya
DOI:10.2174/2211352517666181122130101

Structure-Activity Relationship of Dicoumarol Derivatives as anti- Staphylococcus aureus (Staph Infection) Agents open Access plus

Volume: 17   Issue: 2
Pp: 93-98
Nidaa Rasheed*, Natalie J. Galant and Imre G. Csizmadia
DOI:10.2174/2211352516666181112125458

Pharmacological Exploitation of Non-Steroidal Anti-inflammatory Drugs as Potential Sources of Novel Antibacterial Agents open Access plus

Volume: 17   Issue: 2
Pp: 81-92
Ebrahim M. Yimer*, Ousman A. Mohammed and Seid I. Mohammedseid
DOI:10.2174/2211352516666181008114542

Sonic Stimulation and Low Power Microwave Radiation Can Modulate Bacterial Virulence Towards Caenorhabditis elegans open Access plus

Volume: 17   Issue: 2
Pp: 150-162
Priya Patel, Hiteshi Patel, Dhara Vekariya, Chinmayi Joshi, Pooja Patel, Steven Muskal and Vijay Kothari*
DOI:10.2174/2211352516666181102150049

New Trypanosoma cruzi Trypanothione Reductase Inhibitors Identification using the Virtual Screening in Database of Nucleus Bioassay, Biosynthesis and Ecophysiology (NuBBE) open Access plus

Volume: 17   Issue: 2
Pp: 138-149
Nelcí do C. Santos, Vinícius G. da Paixão and Samuel S. da Rocha Pita*
DOI:10.2174/2211352516666180928130031

Prophylactic and Therapeutic Treatments' Effect of Moringa Oleifera Methanol Extract on Cryptosporidium Infection in Immunosuppressed Mice open Access plus

Volume: 17   Issue: 2
Pp: 130-137
Nagwa M. El-Sayed* and Ghada M. Fathy
DOI:10.2174/2211352517666181221094420

Synthesis of Some 5-(substituted benzylidene-2, 4-dioxothiazolidin-3-yl) benzoic Acid Derivatives by Conventional and Microwave-assisted Methods and Evaluation of their Potential as Antimicrobial Agents open Access plus

Volume: 17   Issue: 2
Pp: 115-129
Karuna S. Shukla, Shailendra Pandey and Pooja Chawla*
DOI:10.2174/2211352516666181024151213

Synthesis and Evaluation of 3-(1,3-dioxoisoindolin-2-yl)-N-substituted Phenyl Benzamide Analogues as HIV Integrase Strand Transfer Inhibitors open Access plus

Volume: 17   Issue: 2
Pp: 105-114
Pankaj Wadhwa*, Priti Jain, Arpit Patel, Shantanu Shinde and Hemant R. Jadhav
DOI:10.2174/2211352516666181102121920

Anti-mitotic Activity of the Benzothiazole-pyrazole Hybrid Derivatives open Access plus

Volume: 17   Issue: 1
Pp: 66-73
M. Bhat*, S.L. Belagali, N.K.H. Kumar and S. Jagannath
DOI:10.2174/2211352516666180914101758

Design, Synthesis and Biological Profiling of Novel Phenothiazine Derivatives as Potent Antitubercular Agents open Access plus

Volume: 17   Issue: 1
Pp: 50-65
Satheeshkumar Sellamuthu, Ashok Kumar, Gopal Nath and Sushil Kumar Singh*
DOI:10.2174/2211352516666180730121013

Comparison of Minimum Inhibitory Concentration (MIC) value of statin drugs: A Systematic Review open Access plus

Volume: 17   Issue: 1
Pp: 4-19
Meenakshi Gupta and Anoop Kumar*
DOI:10.2174/2211352516666180629124433

Modeling and Statistical Optimization of Culture Conditions for Improvement of Antifungal Compounds Production by Streptomyces albidoflavus S19 Strain of Wastewater Origin open Access plus

Volume: 17   Issue: 1
Pp: 39-49
S. Souagui*, W. Djoudi, H. Boudries, M. Béchet, V. Leclére and M. Kecha
DOI:10.2174/2211352516666180813102424

Novel Diazenyl Containing Phenyl Styryl Ketone Derivatives As Antimicrobial Agents open Access plus

Volume: 17   Issue: 1
Pp: 28-38
L. Sivasankerreddy*, B. Nagamani, T. Rajkumar, M.S. Babu, N.Y. Subbaiah, M.S. Harika and R. Nageswarao
DOI:10.2174/2211352516666180927111546

Synthesis, Screening and Docking Analysis of Novel Benzimidazolium and Benzotriazolium Compounds as Potent Anti Tubercular Agents open Access plus

Volume: 17   Issue: 1
Pp: 20-27
Padma Vijaya Sangeeta Guruvelli, Pranita Wagmare, Bhaskar C. Harinath, Risy Namratha Jamullamudi, Purna Nagasree Kurre and Murali Krishna Kumar Muthyala*
DOI:10.2174/2211352516666180810101327

Antibacterial, Antifungal and Anti-tubercular Activities of Chloroform Fraction of the Leaf Extract of Irvingia Gabonensis (African Bush Mango) open Access plus

Volume: 17  
Pp: 1-6
Ifedolapo O. Olanrewaju*, Raphael C. Mordi and JohnBull O. Echeme
DOI:10.2174/2211352517666181122125411

Tetrahydrocarbazoles as Novel Class of DNA Biosynthesis Inhibitors in Bacteria open Access plus

Volume: 17  
Pp: 1-6
Yan A. Ivanenkov*, Ilya A. Osterman, Ekaterina S. Komarova, Alexey A. Bogdanov, Petr V. Sergiev, Olga A. Dontsova, Alina A. Sofronova*, Victor A. Terentiev, Gleb I. Filkov, Renat S. Yamidanov, Alexander G. Majouga, Dmitry S. Bezrukov, Ekaterina V. Deyneka and Dmitry A. Skvortsov
DOI:10.2174/2211352517666181218155259

Antimicrobial Activity of Some Novel 1-(3-(4-Chlorophenylimino)-3,4- dihydroquinoxalin-2-yl)-3-substituted phenyl-1H-pyrazole-4-carbaldehyde open Access plus

Volume: 17  
Pp: 1-7
D. Visagaperumal* and Vineeth Chandy
DOI:10.2174/2211352517666190117143604

Novel Strategies and Pharmaceutical Agents for the Treatment of Leishmaniasis: A Review open Access plus

Volume: 17  
Pp: 1-12
Mohammad Ali Nilforoushzadeh, Maryam Heidari-Kharaji*, Mehrak Zare, Elham Torkamaniha and Sima Rafati
DOI:10.2174/2211352517666190123113843

Telfairia Occidentalis Potentiates the Antiplasmodial Activity of Artemisinins and Amodiaquine Combination Therapy open Access plus

Volume: 17  
Pp: 1-8
Aniekan S. Ebong*, Olorunfemi A. Eseyin, Emmanuel E. Iweh , Jude E. Okokon , Victor U. Anah, Emmanuel E. Attih and Goodnews E. Charles
DOI:10.2174/2211352517666190206160812

Effect of Polypropylene Imine Nanocomposite on Gram-Positive and Gram-Negative Bacteria open Access plus

Volume: 17  
Pp: 1-6
Bashir Mohammadpour*, Mohammad Amin Boshagh, Bagher Hayati, Leila Farhadi, Hajar Kashefi and Himen Salimizand
DOI:10.2174/2211352517666190215114534

In Silico (3D-QSAR) Design, Study, Synthesis and Anti-tubercular Evaluation of Pyrazolo-Pyrimidine Derivatives open Access plus

Volume: 17  
Pp: 1-9
Pratiksha Chhatbar, Kaushik Pambhar, Vijay Khedkar, Anamik Shah and Ranjan Khunt*
DOI:10.2174/2211352517666190225143923

Assessment of Efficacy and Safety of Clindamycin Against Methicillin- Resistant Staphylococcus aureus (MRSA) Infected Subcutaneous Abscess Model open Access plus

Volume: 17  
Pp: 1-8
Lalitha Vivekanandan*, Hajasherief Sheik, Sengottuvelu Singaravel and Sivakumar Thangavel
DOI:10.2174/2211352517666190301142421

Synthesis of piperidine-4-one Derivative Containing Dipeptides: An Acetyl cholinesterase and β-secretase Inhibitor open Access plus

Volume: 17  
Pp: 1-9
Parasuraman Pavadai*, Suresh Ramalingam, Theivendren Panneerselvam, Selvaraj Kunjiappan, Pandurangan Perumal, Vasudevan Mani, Govindaraj Saravanan, Veerachamy Alagarsamy and Damodar Nayak Ammunje
DOI:10.2174/2211352517666190405155505

Synthesis and Biological Activity of Some Aminothiazole Derivatives as Antileishmanial Agents open Access plus

Volume: 17  
Pp: 1-12
Zahra Rezaei*, Bahador Sarkari, Soghra Khabnadideh, Mahbobeh Farjami, Mahsa Mehrjou, Atefeh Yazdi, Elham Riazimontazer and Mohammad Fararouei
DOI:10.2174/2211352517666190527112955

Chemical Composition, Antioxidant, Antibacterial, Cytotoxicity, and Hemolyses Activity of Essential Oils from Flower of Matricariachamomillavar. Chamomilla open Access plus

Volume: 17  
Pp: 1-9
Behnam Mahdavi*, Fereshteh Ghorat, Mahda S. Nasrollahzadeh, Mahmood Hosseyni-Tabar and Hassan Rezaei-Seresht
DOI:10.2174/2211352517666190528114041

Antimicrobial Activity of SPC13, New Antimicrobial Peptide Purified from Scolopendra Polymorpha Venom open Access plus

Volume: 17  
Pp: 1-6
Rodríguez-Alejandro. C. I. and Gutiérrez M.C.*
DOI:10.2174/2211352517666190531110829

Hemolysis, Platelet Aggregation and Antibacterial Activities of Human Antiphospholipid Antibody open Access plus

Volume: 17  
Pp: 1-7
Farzaneh Ahmadi Shapoorabadi, Maryam Sadat Mirbagheri Firoozabad*, Neda Habibi and Giti Emtiazi
DOI:10.2174/2211352517666190613111628

Efficacy of Essential Oil and Hydrosol Extract of Marrubium vulgare on Fungi Responsible for Apples Rot open Access plus

Volume: 17  
Pp: 1-9
Amina Tabet Zatla*, Imane Mami, Mohammed El Amine Dib and Mohammed El Amine Sifi
DOI:10.2174/2211352517666190618105332

Synthesis, Biological Evaluation and Molecular Docking Study of Pyrazole, Pyrazoline Clubbed Pyridine as Potential Antimicrobial Agents open Access plus

Volume: 17  
Pp: 1-9
Nisheeth C Desai*, Darshita V Vaja, Krunalsinh A. Jadeja, Surbhi B. Joshi and Vijay M Khedkar
DOI:10.2174/2211352517666190627144315

Antibacterial Effects of Derivatives of Porphyrin, Naphthalene diimide, Aminophenol and Benzodioxane on Methicillin Resistant Staphylococcus aureus and Neuropathogenic Escherichia coli K1 open Access plus

Volume: 17  
Pp: 1-10
Ruqaiyyah Siddiqui, Ayaz Anwar, Salwa Ali and Naveed Ahmed Khan*
DOI:10.2174/2211352517666190628111232

Design, Synthesis and Antimicrobial Activity of Some Triazine Chalcone Derivatives open Access plus

Volume: 17  
Pp: 1-7
Ravindra Sandipan Shinde*, Satish Ashruba Dake and Rajendra Pundalikrao Pawar
DOI:10.2174/2211352517666190710115111

The Role of Gut Microbiota in Antimicrobial Resistance: A Mini-Review open Access plus

Volume: 17  
Pp: 1-6
Farzaneh Firoozeh and Mohammad Zibaei*
DOI:10.2174/2211352517666190716154013

Cyclo(L-Pro-L-Tyr) from Streptomyces sp. 150: Exploiting in vitro Potential in Controlling Foodborne Pathogens and Phytopathogens open Access plus

Volume: 17  
Pp: 1-9
Atiqur Rahman*, Shah Alam Siddiqui, M. Oliur Rahman and Sun Chul Kang*
DOI:10.2174/2211352517666190716155147

Designing of an Epitope- Based Universal Peptide Vaccine against Highly Conserved Regions in RNA Dependent RNA Polymerase Protein of Human Marburg Virus: A Computational Assay open Access plus

Volume: 17  
Pp: 1-12
S. M. Neaz Mahmud, Md. Mahbubur Rahman, Antora Kar, Nasreen Jahan and Md. Arif Khan*
DOI:10.2174/2211352517666190717143949

Polyaminosteroid Analogues as Potent Antibacterial Agents Against Mupirocin- Resistant Staphylococcus Aureus Strains open Access plus

Volume: 17  
Pp: 1-6
Adèle Sakr, Frédéric Laurent, Jean Michel Brunel, Tania Nawfal Dagher, Olivier Blin and Jean Marc Rolain *
DOI:10.2174/2211352517666190723092347

Phosphonate Derivatives of 3,5-bis(arylidene)-4-piperidone: Synthesis and Biological Evaluation open Access plus

Volume: 17  
Pp: 1-10
Shweta Mishra, Debashree Das, Adarsh Sahu, Shailendra Patil, Ram Kishore Agrawal and Asmita Gajbhiye*
DOI:10.2174/2211352517666190820143735

Synthesis, Biological Evaluation, QSAR, Molecular Docking and ADMET Studies of N-aryl/N,N-dimethyl Substituted Sulphonamide Derivatives open Access plus

Volume: 17  
Pp: 1-10
Samridhi Thakral and Vikramjeet Singh*
DOI:10.2174/2211352517666190902130014

Silica gel Supported Boric tri-Sulfuric Anhydride (SiO2-BTSA): An Efficient Catalytic System for the Synthesis of Phloroglucide Analogs as Antimicrobial Agents open Access plus

Volume: 17  
Pp: 1-10
Rahele Bargebid, Ali Khalafi-Nezhad, Kamiar Zomorodian, Mahkameh Moradi and Soghra Khabnadideh*
DOI:10.2174/2211352517666190902142915

Essential Oil Composition and Anti-scabies Potential of Amomum subulatum Roxb. Leaves open Access plus

Volume: 17  
Pp: 1-7
Bharat Sharma, Neeru Vasudeva* and Sunil Sharma
DOI:10.2174/2211352517666190919143631

Studies on X-Ray Diffraction, Thermogravimetric Stability, Antibacterial- Antifungal Activity of Fe(II), Ni(II), Cu(II) Metal Chloroquine Complexes Against Bacterial Strains and Fungal Spore open Access plus

Volume: 17  
Pp: 1-13
Mukesh Shankarrao Kadam*, Sachin Atmaram Khiste, Satish Ashruba Dake and Bhimrao Chintamanrao Khade
DOI:10.2174/2211352517666191021090630

Synthetic Methods and Antimicrobial Perspective of Pyrazole Derivatives: An Insight open Access plus

Volume: 17  
Pp: 1-17
Harish Kumar, Kushal Kumar Bansal and Anju Goyal*
DOI:10.2174/2211352517666191022103831

Synthesis and SAR Evaluation of Mercapto Triazolobenzothiazole Derivatives as Anti-tuberculosis Agents open Access plus

Volume: 17  
Pp: 1-13
Mamatha S. V*, S. L. Belagali and Mahesh Bhat
DOI:10.2174/2211352517666191204095558

The in vitro Antiviral Mechanisms of Stronger Neo-Minophafen C, an Established Formulation of Compound Glycyrrhizin open Access plus

Volume: 16   Issue: 2
Pp: 136-143
Chi Zhang, Qi-Jie Li, Yi-Li Wang, Jie Chen, Chun-Yan Lv, Wei-Wei Liu, Li Chen, Jia-Yue He, De-Yu Jiang, Xiu-Wen Xia and Wei-Jun Ding*
DOI:10.2174/2211352516666180619142745

Sulfonamides as Inhibitors of Leishmania – Potential New Treatments for Leishmaniasis open Access plus

Volume: 15   Issue: 1
Pp: 57-62
Jade Katinas*, Rachel Epplin, Christopher Hamaker and Marjorie A. Jones
DOI:10.2174/2211352515666170216143401