Abstract
The present review contains a representative sampling from the last 10 years on the synthesis of biologically interesting compounds, prepared by the use of the 1,3-dipolar cycloaddition and Diels-Alder reactions, that have been eventually sequenced into cascade processes to assemble heterocyclic molecules. The important role of click chemistry for the synthesis of bio-inspired compounds have been also outlined.
Keywords: Cycloaddition Methodology, Diels-Alder reactions, heterocyclic molecules, synthesis
Current Organic Chemistry
Title: Cycloaddition Methodology: A Useful Entry Towards Biologically Active Heterocycles
Volume: 13 Issue: 5
Author(s): Ugo Chiacchio, Albert Padwa and Giovanni Romeo
Affiliation:
Keywords: Cycloaddition Methodology, Diels-Alder reactions, heterocyclic molecules, synthesis
Abstract: The present review contains a representative sampling from the last 10 years on the synthesis of biologically interesting compounds, prepared by the use of the 1,3-dipolar cycloaddition and Diels-Alder reactions, that have been eventually sequenced into cascade processes to assemble heterocyclic molecules. The important role of click chemistry for the synthesis of bio-inspired compounds have been also outlined.
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Cite this article as:
Chiacchio Ugo, Padwa Albert and Romeo Giovanni, Cycloaddition Methodology: A Useful Entry Towards Biologically Active Heterocycles, Current Organic Chemistry 2009; 13 (5) . https://dx.doi.org/10.2174/138527209787582268
DOI https://dx.doi.org/10.2174/138527209787582268 |
Print ISSN 1385-2728 |
Publisher Name Bentham Science Publisher |
Online ISSN 1875-5348 |
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