Letters in Drug Design & Discovery

Editor-in-Chief
K. Kuca
University of Hradec Kralove
Hradec Kralove
Czech Republic

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Volume:8   Issue: 10
Pp: i-v

DOI: 10.2174/157018011797655313

MGBG in Combined Anticancer Chemotherapy

Volume:8   Issue: 10
Pp: 897-903
R. F. Goncalves, G. Kriechammer and M. P.M. Marques
DOI: 10.2174/157018011797655197

Titanocene Y and Vanadocene Y: Platinum Resistance-Breaking Cytotoxic and DNA-Targeting Anticancer Drug Candidates

Volume:8   Issue: 10
Pp: 904-910
Ralf A. Hilger, Dennis Alex, Anthony Deally, Brendan Gleeson and Matthias Tacke
DOI: 10.2174/157018011797655241

Synthesis and Biological Evaluation of Licofelone Derivatives as Anticancer and Anti-inflammatory Agents

Volume:8   Issue: 10
Pp: 911-917
Wukun Liu, Jinpei Zhou, Huibin Zhang, Hai Qian, Jiahan Yin, Kerstin Bensdorf and Ronald Gust
DOI: 10.2174/157018011797655223

3D-QSAR Studies of VEGFR-2 Kinase Inhibitors Based on Docking

Volume:8   Issue: 10
Pp: 926-942
Xiaoping Jiang, Guangchuan Ou, Depeng Yan, Min Zhang and Xianyou Yuan
DOI: 10.2174/157018011797655296

Synthesis and Preliminary Screening of Novel A- and D-Ring Modified Steroids as Aromatase Inhibitors

Volume:8   Issue: 10
Pp: 943-950
Mange Ram Yadav, Prafulla M. Sabale, Rajani Giridhar, Dharmendra Baria, Christina Zimmer and Rolf W. Hartmann
DOI: 10.2174/157018011797655322

A Novel Bromomelatonin Derivative Suppresses Apoptosis with Regulating the Expression of Bcl-2 Family Genes

Volume:8   Issue: 10
Pp: 951-956
Yoshikazu Mikami, Masanori Somei, Eri Watanabe, Nobukazu Watanabe, Tomihisa Takahashi and Masaki J. Honda
DOI: 10.2174/157018011797655287

Synthesis of Cinnamide Dimers as Potential Antibacterial and Antifungal Agents

Volume:8   Issue: 10
Pp: 957-965
Ahmed Kamal, G. Ramakrishna, P. Raju, A. V. Subba Rao, Joveeta Joseph, B. Siddhardha and U. S.N. Murty
DOI: 10.2174/157018011797655205

Novel Clarithromycin Analogs with C-4” 2-arylbenzimidazolyl Bishydrazide Side Chain: Synthesis and Antibacterial Evaluation

Volume:8   Issue: 10
Pp: 966-971
Yunkun Qi, Ruixin Ma, Xin Li, Yue Hu, Siti Ma, Chao Cong, Xiaodong Ma, Wenping Cui and Shutao Ma
DOI: 10.2174/157018011797655269

Synthesis and Antibacterial Activity of 6-Substituted Anacardic Acid Derivatives

Volume:8   Issue: 10
Pp: 972-979
Subhakara Reddy Nallamilli, Ravi Kumar V, Himabindu V, B. Ram and Srinivas Rao Aalapati
DOI: 10.2174/157018011797655278

Antimicrobial Efficacy of Metal-Barbiturate Conjugates Against Pathogenic Strains of Escherichia coli and Staphylococcus aureus

Volume:8   Issue: 10
Pp: 980-987
Ashfaq Mahmood Qureshi, Mehmood Qadir, Abdul Rauf, Muhammad Idrees, Siara Mumtaz, Muhammad Najam-ul-Haq, Muhammad Ismail, Muhammad Athar, Rashid Khushal, Sara Riaz and Habib Bokhari
DOI: 10.2174/157018011797655232

Synthesis of 2-methyl-3-(2-(piperazin-1-yl)ethyl)-6,7,8,9-tetrahydro-4Hpyrido[ 1,2-a]pyrimidin-4-one Derivatives as Antimicrobial Agents

Volume:8   Issue: 10
Pp: 988-995
Byregowda Krishnamurthy, Kambappa Vinaya, Doddakunche S. Prasanna, Byregowda Raghava and Kanchugarakoppal S. Rangappa
DOI: 10.2174/157018011797655304

Molecular Mapping and Docking Interactions for Selective Anti-Fertility Potency of Estrogen Analogs

Volume:8   Issue: 10
Pp: 996-1003
Ria Pal, Md Ataul Islam, Tabassum Hossain and Achintya Saha
DOI: 10.2174/157018011797655214