Letters in Drug Design & Discovery

Editor-in-Chief:

George Perry
University of Texas
San Antonio, TX
USA

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Volume:7   Issue:6
Pp: i-iv

DOI: 10.2174/157018010791306506

Synthesis and Evaluation of Estradiol Derivatives as Anti-Breast Cancer Agents

Volume:7   Issue:6
Pp: 389-394
John S. Cooperwood, Jesse Edwards, Musiliyu Musa, Devora Simmons, Abdul D. Mian, Kwon-kyun Park and Zhongliang Wan
DOI: 10.2174/157018010791306551

Self-Organizing Molecular Field Analysis on Pyridazine Analogues as Protein Tyrosine Phosphatase 1B (PTP 1B) Inhibitors

Volume:7   Issue:6
Pp: 395-401
Suresh Thareja, Saurabh Aggarwal, Tilak Raj Bhardwaj and Manoj Kumar
DOI: 10.2174/157018010791306605

Evaluation of Novel 7-(hetero)aryl-substituted Pyrazolo[1, 5-a]pyrimidines as Phosphodiesterase-4 Inhibitors

Volume:7   Issue:6
Pp: 402-408
Arumugam Kodimuthali, Rajesh Gupta, Kishore Venkata Laxmi Parsa, Padala Lakshmi Prasunamba and Manojit Pal
DOI: 10.2174/157018010791306542

Assessing Drugs for their Cardio-Toxicity

Volume:7   Issue:6
Pp: 409-414
Anwar Rayan, Mizied Falah, Jamal Raiyn, Hafiz Mawassi and Nur-Eldin Raiyn
DOI: 10.2174/157018010791306515

Design, Synthesis and Biological Evaluation of Benzopyran Derivatives as KATP Channel Openers

Volume:7   Issue:6
Pp: 415-420
Jinpei Zhou, Hai Qian, Huibin Zhang, Hui Gao, Wenlong Huang, Xiaoyun Zhu, Shuaijian Ni and Chuntao Zhang
DOI: 10.2174/157018010791306560

Design and Synthesis of Novel 1,3-Dioxane-2-carboxylic Acid Derivatives as PPARα/γ Dual Agonists

Volume:7   Issue:6
Pp: 421-429
Harikishore Pingali, Mukul Jain, Shailesh Shah, Pankaj Makadia, Pandurang Zaware, Jeevankumar Jamili, Kalapatapu V.V.M. Sairam, Pravin Patil, Dinesh Suthar, Suresh Giri, Harilal Patel and Pankaj Patel
DOI: 10.2174/157018010791306533

Application of Molecular Topology to the Search of Novel NSAIDs: Experimental Validation of Activity

Volume:7   Issue:6
Pp: 438-445
Maria Galvez-Llompart, Rosa M. Giner, Maria C. Recio, Sanzio Candeletti and Ramon Garcia-Domenech
DOI: 10.2174/157018010791306597

Synthesis and Biological Evaluation of Novel Bioisosteric Analogues of Dimebon™

Volume:7   Issue:6
Pp: 446-451
Alexandre Vasilevich Ivachtchenko, Eugene Borisovich Frolov, Oleg Dmitrievich Mitkin, Sergey Evgenevich Tkachenko and Alexandre Khvat
DOI: 10.2174/157018010791306579

New Limonene-Hybrid Derivatives with Anti-T. cruzi Activity

Volume:7   Issue:6
Pp: 452-460
G. Alvarez, A. Gerpe, D. Benitez, F. Garibotto, S. Zacchino, C. S. Graebin, R. Gomes da Rosa, V. L. Eifler-Lima, M. Gonzalez and H. Cerecetto
DOI: 10.2174/157018010791306524

Synthesis and Anticoccidial Activity of 3-(2-(1-methoxynaphthalen-2-yl)-2-oxoethyl) Quinazolinone Derivatives

Volume:7   Issue:6
Pp: 471-475
Yuanyuan Zhang, Guangmin Chen, Yabiao Weng, Renliang Li, Yuliang Wang and Yuzhong Wang
DOI: 10.2174/157018010791306498