Letters in Drug Design & Discovery

Editor-in-Chief
K. Kuca
University of Hradec Kralove
Hradec Kralove
Czech Republic

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Structure-Based Drug Design of Peptide Mimetics Containing Large P3 Moieties as Inhibitors of Factor VIIa

Volume:6   Issue: 2
Pp: 86-92
Takuya Shiraishi, Shojiro Kadono, Masayuki Haramura, Hirofumi Kodama, Yoshiyuki Ono, Hitoshi Iikura, Tohru Esaki, Takaki Koga, Kunihiro Hattori, Yoshiaki Watanabe, Akihisa Sakamoto, Kazutaka Yoshihashi, Takehisa Kitazawa, Keiko Esaki, Masateru Ohta, Haruhiko Sato and Toshiro Kozono
DOI: 10.2174/157018009787582606

Novel N-Substituted Thiazolidinones as Proton Pump Inhibitors and Potent Anti-Ulcer Agents: SAR Study

Volume:6   Issue: 2
Pp: 101-106
S. Chandrappa, K. Vinaya, B. M. Srikanta, C.S. Ananda Kumar, N. R. Thimmegowda, S. R. Ranganatha, Shylaja M. Dharmesh and K. S. Rangappa
DOI: 10.2174/157018009787582697

Synthesis of Substituted 1H-Pyrrol-2(5H)-ones and 2(5H)-Furanones as Inhibitors of P. aeruginosa Biofilm

Volume:6   Issue: 2
Pp: 107-113
Jia-Liang Guo, Bing-Zhou Li, Wei-Min Chen, Ping-Hua Sun and Yuqiang Wang
DOI: 10.2174/157018009787582642

Physical Stability of PLGA Microparticles for DNA Encapsulation

Volume:6   Issue: 2
Pp: 125-128
Itziar Migueliz, Sonsoles Diez, Gemma Navarro and Conchita Tros de ILarduya
DOI: 10.2174/157018009787582679

A Novel Synthesis Method of Apogossypolone and its Antitumor Activity

Volume:6   Issue: 2
Pp: 129-132
Yonghua Zhan and Guangfeng Jia
DOI: 10.2174/157018009787582589

Synthesis and Antiproliferative Activity of Coumarin-Estrogen Conjugates against Breast Cancer Cell Lines

Volume:6   Issue: 2
Pp: 133-138
Musiliyu A. Musa, M. Omar F. Khan and John S. Cooperwood
DOI: 10.2174/157018009787582624

Presentation of the β -Carboxamidophosphonate Arrangement in Substrate Structures Targeting HIV-1 PR

Volume:6   Issue: 2
Pp: 139-145
N. J. Wardle, H. R. Hudson, R. W. Matthews, C. Nunn, C. Vella and S.W. A. Bligh
DOI: 10.2174/157018009787582660

Synthesis and In Vitro Antimicrobial Activity of Medicinally Important Novel N-alkyl, N-aryl and Urea Derivatives of 1-benzhydryl Piperizine: A Structure-Activity Relationship Study

Volume:6   Issue: 2
Pp: 146-154
Channapillekoppal Siddegowda Ananda Kumar, Karunakara Murthy, Marlinganadoddi Panchegowda Sadashiva, Mallappanahally Kambappa Vinaya, Naraganahalli Ramegowda Thimmegowda, Salekoppal Boregowda Benaka Prasad, Siddappa Chandrappa and Kanchugarakoppal Subbegowda Rangappa
DOI: 10.2174/157018009787582570

Complex of Nifedipine with Glycyrrhizic Acid as a Novel Water-Soluble Antihypertensive and Antiarrhythmic Agent

Volume:6   Issue: 2
Pp: 155-158
T. G. Tolstikova, M. V. Khvostov, A. O. Bryzgalov, A. V. Dushkin and E. S. Meteleva
DOI: 10.2174/157018009787582688

3-Aminosterol Compounds as a New Class of Anti-Malarial Agents against Chloroquine-Susceptible and -Resistant Plasmodium falciparum

Volume:6   Issue: 2
Pp: 163-166
Chanaz Salmi, Celine Loncle, Nicolas Vidal, Christophe Rogier, Yves Letourneux, Bruno Pradines and Jean Michel Brunel
DOI: 10.2174/157018009787582633