Letters in Drug Design & Discovery

Editor-in-Chief
K. Kuca
University of Hradec Kralove
Hradec Kralove
Czech Republic

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Meet Our Editor-in-Chief free to download

Volume:17   Issue: 1
Pp: 1-1
Kamil Kuca
DOI: 10.2174/157018081701191211104947



Preface free to download

Volume:17   Issue: 1
Pp: 2-2
Kamil Kuca
DOI: 10.2174/157018081701191211105210



Targeting Inflammation with Conjugated Cinnamic Amides, Ethers and Esters

Volume:17   Issue: 1
Pp: 3-11
Ioannis Fotopoulos, Eleni Pontiki and Dimitra Hadjipavlou Litina*
DOI: 10.2174/1570180816666181129125511



Synthesis and SAR Study of Simple Aryl Oximes and Nitrofuranyl Derivatives with Potent Activity Against Mycobacterium tuberculosis

Volume:17   Issue: 1
Pp: 12-20
Cristiane França da Costa, Marcus Vinicius Nora de Souza*, Maria Cristina da Silva Lourenço, Elaine Soares Coimbra, Guilherme da Silva Lourenço Carvalho, James Wardell, Stephane Lima Calixto and Juliana da Trindade Granato
DOI: 10.2174/1570180816666181227115738



Melatonin Ameliorates Radiation-induced Sciatic Nerve Injury

Volume:17   Issue: 1
Pp: 21-30
Dheyauldeen Shabeeb*, Ahmed Eleojo Musa, Mansoor Keshavarz, Gholamreza Hassanzadeh, Mohammed Reza Hadian, Azin Nowrouzi, Alireza Shirazi* and Masoud Najafi
DOI: 10.2174/1570180816666190617160434



Identifying the Structural Features of Diphenyl Ether Analogues for InhA Inhibition: A 2D and 3D QSAR Based Study

Volume:17   Issue: 1
Pp: 31-47
Ashutosh Prasad Tiwari, Varadaraj Bhat Giliyar*, Gurypur Gautham Shenoy and Vandana Kalwaja Eshwara
DOI: 10.2174/1570180816666190611153933



Antimicrobial Activity, Antioxidant Properties and Phytochemical Screening of Aesculus hippocastanum Mother Tincture against Food-borne Bacteria

Volume:17   Issue: 1
Pp: 48-56
Maria Grazia Bonomo*, Caterina Cafaro, Daniela Russo, Luana Calabrone, Luigi Milella, Carmela Saturnino, Anna Capasso and Giovanni Salzano
DOI: 10.2174/1570180816666181108114115



Synthesis and Analgesic Activity of Monoterpenoid Aldehyde-derived Hydro-2H-chromeneols

Volume:17   Issue: 1
Pp: 68-78
Irina Il'ina*, Ekaterina Morozova, Dina Korсhagina, Konstantin Volсho, Tat'yana Tolstikova and Nariman Salakhutdinov
DOI: 10.2174/1570180816666181114131220



One-pot Synthesis of Betulin Triterpenoid Quaternized Pyridine Derivatives and their Antimicrobial Activity

Volume:17   Issue: 1
Pp: 79-84
Elvira Rifovna Shakurova, Darina Alexandrovna Pozdnyakova, Elena Valeryevna Tretyakova and Lyudmila Vyacheslavovna Parfenova*
DOI: 10.2174/1570180816666181217123629



Synthesis of Piperidine Conjugated Dihydroquinazolin-4(1H)-ones and their Antiproliferative Activity, Molecular Docking Studies and DFT Calculations

Volume:17   Issue: 1
Pp: 85-93
Kereyagalahally Honneshappa Narasimhamurthy, Chandra, Toreshettahally Ramesh Swaroop, Swamy Jagadish and Kanchugarakoppal Subbegowda Rangappa*
DOI: 10.2174/1570180816666190613120349



Synthesis and Antimicrobial Activity of Thiohydantoins Obtained from L-Amino Acids

Volume:17   Issue: 1
Pp: 94-102
Priscila Goes Camargo de Carvalho, Jhonatan Macedo Ribeiro, Renata Perugini Biasi Garbin, Gerson Nakazato, Sueli Fumie Yamada Ogatta, Ângelo de Fátima, Marcelle de Lima Ferreira Bispo and Fernando Macedo*
DOI: 10.2174/1570180816666181212153011