Letters in Drug Design & Discovery

Editor-in-Chief
K. Kuca
University of Hradec Kralove
Hradec Kralove
Czech Republic

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Volume:16   Issue: 4
Pp: 371-371
Bruno Rizzuti
DOI: 10.2174/157018081604190220100304



Benzothiazol Clubbed Imidazol-4-ones as Anti-fungal, Anti-tubercular and Anti-HIV-1 Agents: Their Synthesis and Molecular Docking Study

Volume:16   Issue: 4
Pp: 382-391
Navin B. Patel*, Asif R. Shaikh, Vatsal M. Patel, Edgar E. Lara-Ramirez and Gildardo Rivera
DOI: 10.2174/1570180815666180712150050



Synthesis, Molecular Modelling and Antibacterial Activity Against Helicobacter pylori of Novel Diflunisal Derivatives as Urease Enzyme Inhibitors

Volume:16   Issue: 4
Pp: 392-400
Göknil Pelin Coşkun, Teodora Djikic, Sadık Kalaycı, Kemal Yelekçi, Fikrettin Şahin and Ş. Güniz Küçükgüzel*
DOI: 10.2174/1570180815666180627130208



Synthesis of 3-Arylindazole-1-acetic Acids and In Vitro Study of Potential Antibacterial Effect

Volume:16   Issue: 4
Pp: 401-407
Fauzia Anjum Chattha, Samina Kousar, Mehr-un-Nisa and Munawar Ali Munawar*
DOI: 10.2174/1570180815666180702152259



Anti-Microbial and Free Radical Scavenging Activities of Nigella Sativa Colloidal-Emulgel

Volume:16   Issue: 4
Pp: 408-416
Ahmad M. Eid*, Nidal A. Jaradat, Nagib A. Elmarzugi, Raed Alkowni, Fatima Hussen, Laila A. Ayyash, Maher Sawafta and Hadeel Danaa
DOI: 10.2174/1570180815666180620150922



Virtual Screening, Molecular Modelling and Biochemical Studies to Exploit PF14_0660 as a Target to Identify Novel Anti-malarials

Volume:16   Issue: 4
Pp: 417-426
Vimee Raturi, Kumar Abhishek, Subhashis Jana, Subhendu Sekhar Bag and Vishal Trivedi*
DOI: 10.2174/1570180815666180727121200



Evaluation of the in vitro Antitumor Activity of Nanostructured Cyclotides in Polymers of Eudragit® L 100-55 and RS 30 D

Volume:16   Issue: 4
Pp: 437-445
Osmar N. Silva, Michelle F.S. Pinto, Juliane F.C. Viana, Camila G. Freitas, Isabel C.M. Fensterseifer, David J. Craik and Octavio L. Franco*
DOI: 10.2174/1570180815666180801115526



Design and Synthesis of Novel Thiosemicarbazones as Potent Anti-breast Cancer Agents open access plus

Volume:16   Issue: 4
Pp: 446-452
Mashooq Ahmad Bhat*, M. Al-Tahhan, Mohamed A. Al-Omar, Ahmed M. Naglah and Abdullah Al-Dhfyan
DOI: 10.2174/1570180815666181008100944



QSAR Studies on Thiazole Derivatives as HCV NS5A Inhibitors via CoMFA and CoMSIA Methods

Volume:16   Issue: 4
Pp: 453-460
Jiayu Li, Wenyue Tian, Diaohui Gao, Yuying Li, Yiqun Chang, Jun Xu, Junxia Zheng* and Pinghua Sun*
DOI: 10.2174/1570180815666180702153529



2-Acryloyl-4,5-methylenedioxyphenol: A Small Molecule Endowed with Antidermatophytic Activity

Volume:16   Issue: 4
Pp: 461-466
Marco Zuccolo, Sabrina Dallavalle*, Raffaella Cincinelli, Luce Mattio, Stefania Mazzini, Michelandrea De Cesare and Loana Musso
DOI: 10.2174/1570180815666180803115347



Theoretical Coupling and Stability of Boronic Acid Adducts with Catecholamines

Volume:16   Issue: 4
Pp: 467-475
Eugeniy Demianenko, Alexey Rayevsky, Marvin A. Soriano-Ursúa* and José G. Trujillo-Ferrara*
DOI: 10.2174/1570180815666180710101604