Letters in Drug Design & Discovery

Editor-in-Chief:

George Perry
University of Texas
San Antonio, TX
USA

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Volume:16   Issue:3
Pp: 237-237
Yiyun Cheng
DOI: 10.2174/157018081603190108093716



A Study on the Synthesis of Risedronic Acid: The Role of an Ionic Liquid Additive open access plus

Volume:16   Issue:3
Pp: 238-244
Dávid Illés Nagy, Alajos Grün, Júlia Sinkovicz, Sándor Garadnay, István Greiner and György Keglevich*
DOI: 10.2174/1570180815666180626122630



Total Synthesis and Antibacterial Screening of (±)-6,8-Dihydroxy-3- undecyl-3,4-dihydroisochromen-1-one: A Structural Analogue of Metabolites from Ononis natrix

Volume:16   Issue:3
Pp: 245-248
Hummera Rafique*, Aamer Saeed, Ehsan Ullah Mughal, Muhammad Naveed Zafar, Amara Mumtaz, Naghmana Kausar and Kiran Hina
DOI: 10.2174/1570180815666180502114402



Green Synthesis, Characterization, DPPH and Ferrous Ion-chelating (FIC) Activity of Tetrakis-Schiff’s Bases of Terephthalaldehyde

Volume:16   Issue:3
Pp: 249-255
Momin Khan*, Umar Ali, Anis Ur Rahman, Muhammad Ibrahim, Abdul Hameed, Muhammad Asif, Zahid Hussain, Kanwal, Khalid Mohammed Khan, Shahnaz Perveen and Munir ur Rehman
DOI: 10.2174/1570180815666180531101404



Coumarinyl Aryl/Alkyl Sulfonates with Dual Potential: Alkaline Phosphatase and ROS Inhibitory Activities: In-Silico Molecular Modeling and ADME Evaluation

Volume:16   Issue:3
Pp: 256-272
Uzma Salar, Khalid Mohammed Khan*, Syeda Abida Ejaz, Abdul Hameed, Mariya al-Rashida, Shahnaz Perveen, Muhammad Nawaz Tahir, Jamshed Iqbal* and Muhammad Taha
DOI: 10.2174/1570180815666180327125738



Cytotoxicity and Molecular Targeting Study of Novel 2-Chloro-3- substituted Quinoline Derivatives as Antitumor Agents

Volume:16   Issue:3
Pp: 273-283
Mohammed A.M. Massoud*, Magda A. El-Sayed, Waleed A. Bayoumi and Basem Mansour
DOI: 10.2174/1570180815666180604090924



Assessing the Antimalarial Potentials of Phytochemicals: Virtual Screening, Molecular Dynamics and In-Vitro Investigations

Volume:16   Issue:3
Pp: 291-300
Saumya K. Patel, Mohd Athar, Prakash C. Jha*, Vijay M. Khedkar, Yogesh Jasrai, Himanshu A. Pandya, Linz-buoy George, Hyacinth Highland and Supriya Sharma
DOI: 10.2174/1570180815666180604085626



3D QSAR Based Virtual Screening of Pyrido[1,2-a] Benzimidazoles as Potent Antimalarial Agents

Volume:16   Issue:3
Pp: 301-312
Kalicharan Sharma, Apeksha Srivastava, Pooja Tiwari, Shweta Sharma, Mohammad Shaquiquzzaman, M. Mumtaz Alam and Mymoona Akhter*
DOI: 10.2174/1570180815666180502115147



Synthesis, Structure Elucidation and Biological Activities of Some Novel 4(3H)-Quinazolinones as Anti-Biofilm Agents

Volume:16   Issue:3
Pp: 313-321
Sevda Türk, Sevgi Karakuş*, Abdulilah Ece, Seyhan Ulusoy and Gülgün Bosgelmez-Tınaz
DOI: 10.2174/1570180815666180621101123



Synthesis and Evaluation of Chalcone and its Derivatives as Potential Anticholinergic Agents

Volume:16   Issue:3
Pp: 322-332
Shahzad Murtaza*, Khoula Zubair Mir, Adina Tatheer and Raja Summe Ullah
DOI: 10.2174/1570180815666180523085436



Aurones as New Porcine Pancreatic α-Amylase Inhibitors

Volume:16   Issue:3
Pp: 333-340
Khashayar Roshanzamir, Elaheh Kashani-Amin, Azadeh Ebrahim-Habibi* and Latifeh Navidpour*
DOI: 10.2174/1570180815666180712150600



N-Acetylserotonin vs Melatonin: In-Vitro Controlled Release from Hydrophilic Matrix Tablets

Volume:16   Issue:3
Pp: 347-352
M. Vlachou*, G. Stavrou, A. Siamidi, S. Flitouri, V. Ioannidou and S. Mavrokordopoulos
DOI: 10.2174/1570180815666180404125519



Evaluation of a Series of 9,10-Anthraquinones as Antiplasmodial Agents

Volume:16   Issue:3
Pp: 353-363
Che Puteh Osman*, Nor Hadiani Ismail, Aty Widyawaruyanti, Syahrul Imran, Lidya Tumewu, Chee Yan Choo and Sharinah Ideris
DOI: 10.2174/1570180815666180607085102



Synthesis of 3-furanyl-4,5-dihydroisoxazole Derivatives via Cycloaddition and their Antibacterial Evaluation

Volume:16   Issue:3
Pp: 364-369
Gabriela de Andrade Danin Barbosa, Alcino Palermo de Aguiar*, Erika Martins de Carvalho and Joseli Maria da Rocha Nogueira
DOI: 10.2174/1570180815666180627115606