Letters in Drug Design & Discovery

Editor-in-Chief:

George Perry
University of Texas
San Antonio, TX
USA

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Volume:16   Issue:2
Pp: 101-101
Romeo Romagnoli
DOI: 10.2174/157018081602181116142645



Synthesis and Biological Evaluation of Some Novel Thiophene-bearing Quinazoline Derivatives as EGFR Inhibitors open access plus

Volume:16   Issue:2
Pp: 102-110
Min Zou, Bo Jin, Yanrong Liu, Huiping Chen, Zhuangli Zhang, Changzheng Zhang, Zhihong Zhao and Liyun Zheng*
DOI: 10.2174/1570180815666180803125935



Synthesis and Anticancer Activity of Some 1H-inden-1-one Substituted (Heteroaryl)Acetamide Derivatives

Volume:16   Issue:2
Pp: 111-118
Ahmet Cagri Karaburun, Nalan Gundogdu-Karaburun*, Leyla Yurttas, Ismail Kayagil and Seref Demirayak
DOI: 10.2174/1570180815666180606081042



The Impact of Antioxidants from the Diet on Breast Cancer Cells Monitored by Raman Microspectroscopy

Volume:16   Issue:2
Pp: 127-137
Paula Sofia Coutinho Medeiros, Ana Lúcia Marques Batista de Carvalho*, Cristina Ruano, Juan Carlos Otero and Maria Paula Matos Marques
DOI: 10.2174/1570180815666180502120804



Indolin-2-one Derivatives: Theoretical Studies Aimed at Finding More Potent Aurora B Kinase Inhibitors

Volume:16   Issue:2
Pp: 138-152
Ítalo Antônio Fernandes, Tamiris Maria de Assis, Isael Aparecido Rosa and Elaine Fontes Ferreira da Cunha*
DOI: 10.2174/1570180815666180528090945



QSAR and Docking Studies of DATA Analogues as HIV-1 Reverse Transcriptase Inhibitors

Volume:16   Issue:2
Pp: 153-159
Jianbo Tong*, Shan Lei, Pei Zhan, Shangshang Qin and Yang Wang
DOI: 10.2174/1570180815666180413152636



Synthesis, Antimicrobial Evaluation and In silico Studies of Novel 2,4- disubstituted-1,3-thiazole Derivatives

Volume:16   Issue:2
Pp: 160-173
Mir Mohammad Masood, Mohammad Irfan, Shadab Alam , Phool Hasan, Aarfa Queen, Shifa Shahid, Muhammad Zahid, Amir Azam and Mohammad Abid*
DOI: 10.2174/1570180815666180502120042



Synthesis and Antichlamydial Activity of Novel Phenazines

Volume:16   Issue:2
Pp: 174-181
Xiaofeng Bao, Xiaowei Yu, Chao Xia, Ningjing Yang, Shengju Yang* and Yu Zhao*
DOI: 10.2174/1570180815666180518112952



Synthesis, Cytotoxic Evaluation, and Molecular Docking Studies of N-(7- hydroxy-4-methyl-2-oxoquinolin-1(2H)-yl)acetamide/benzamide Analogues

Volume:16   Issue:2
Pp: 182-193
Mohamed Jawed Ahsan*, Rupesh Kumar Kumawat, Surender Singh Jadav, Mohammed H. Geesi, Mohammed Afroz Bakht, Mohd. Zaheen Hassan, Abdulmalik Bin Saleh Al-Tamimi, Yassine Riadi , Salahuddin, Afzal Hussain, Narayan Murthy Ganta and Habibullah Khalilullah
DOI: 10.2174/1570180815666180501160047



Design, Synthesis and In vitro Cytotoxicity of New 1,2,3-triazol- and Nitrostyrene Hybrids as Potent Anticancer Agents

Volume:16   Issue:2
Pp: 213-219
Zahra Tashrifi, Maryam Mohammadi-khanaposhtani, Mehdi Shafiee Ardestani, Maliheh Safavi, Kurosh Rad-Moghadam*, Morteza Mehrdad, Bagher Larijani and Mohammad Mahdavi*
DOI: 10.2174/1570180815666180427151830



Dual Acting Isatin-heterocyclic Hybrids: Recent Highlights as Promising Pharmacological Agents

Volume:16   Issue:2
Pp: 220-236
Srinubabu Maddela*, Githa Elizabeth Mathew, Della Grace Thomas Parambi, Fakhria Aljoufi and Bijo Mathew*
DOI: 10.2174/1570180815666180516102100