Letters in Drug Design & Discovery

Editor-in-Chief
K. Kuca
University of Hradec Kralove
Hradec Kralove
Czech Republic

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Volume:15   Issue: 6
Pp: 575-575
Adriano Mollica
DOI: 10.2174/157018081506180420152052



Novel Hybrid Molecules of Isoxazole Chalcone Derivatives: Synthesis and Study of in vitro Cytotoxic Activities

Volume:15   Issue: 6
Pp: 576-582
Arunkumar Thiriveedhi*, Ratnakaram Venkata Nadh, Navuluri Srinivasu and Kishore Kaushal
DOI: 10.2174/1570180814666170914121740




Microwave-promoted Synthesis of S-substituted Quinazoline Derivatives using 1,4-dihydroquinazoline-2-thiol

Volume:15   Issue: 6
Pp: 583-589
Satya Karuna Pulakhandam, Naresh Kumar Katari* and Ravi Prakash Reddy Manda
DOI: 10.2174/1570180814666170823160851




1, 2, 4-Oxadiazole Incorporated Ketoprofen Analogues in Search of Safer Non-steroidal Anti-inflammatory Agents: Design, Syntheses, Biological Evaluation and Molecular Docking Studies

Volume:15   Issue: 6
Pp: 590-601
Chanda Ranjan, Jagdish Kumar, Kalicharan Sharma, Mymoona Akhter, Anees A. Siddiqui and Gita Chawla*
DOI: 10.2174/1570180814666170810115134




Synthesis, Antioxidant and Antimicrobial Activities of Metal Complexes of 2-thiouracil-hydroxyquinoline Derivatives

Volume:15   Issue: 6
Pp: 602-611
Apilak Worachartcheewan*, Ratchanok Pingaew, Decha Lekcharoen, Supaluk Prachayasittikul*, Somsak Ruchirawat and Virapong Prachayasittikul
DOI: 10.2174/1570180814666170922163828




Comparative Antioxidant Activity and Structural Feature of Protocatechuic Acid and Phenolic Acid Derivatives by DPPH and Intracellular ROS

Volume:15   Issue: 6
Pp: 612-620
Woong Kim, Beomgi Lee, Jaeyoung Park, Ho-Joong Kim and Hyeonsook Cheong*
DOI: 10.2174/1570180814666171002161302




Microwave Assisted Synthesis and Potent Antimicrobial Activity of Some Novel 1,3-dialkyl-2-arylbenzimidazolium Salts

Volume:15   Issue: 6
Pp: 621-633
Bilge Eren*, Ozge Yilmaz, Gulcin Cetin and Cihan Darcan
DOI: 10.2174/1570180814666170823162419




In Silico Study of Flavonoids as DPP-4 and α-glucosidase Inhibitors

Volume:15   Issue: 6
Pp: 634-642
Jasmin Kaur, Ramit Singla and Vikas Jaitak*
DOI: 10.2174/1570180814666170915162232




A Computational Study of Molecular Interactions and In Vitro Antibacterial Activity of 6-Substituted Quinoline Carboxylic Acid Derivatives as DNA Gyrase Inhibitors

Volume:15   Issue: 6
Pp: 643-653
Sonal Dubey*, Sakshi Bhardwaj, Ekta Singh, Prabitha Prabhakaran and Ayda Cherian
DOI: 10.2174/1570180814666170810114508




Pharmacophore and 3D-QSAR Characterization of Thieno[3,2-d] pyrimidine-6-carboxamides as SIRT-2 Inhibitors

Volume:15   Issue: 6
Pp: 661-670
Neetu Agrawal*, Kamal Shah and Pradeep Mishra
DOI: 10.2174/1570180814666170918145317




Synthesis and Mosquitocidal Activity of a Series of Hydrazone Derivatives against Aedes aegypti

Volume:15   Issue: 6
Pp: 671-677
Mehlika Dilek Altintop*, Nurhayat Tabanca, James J. Becnel, Jeffrey R. Bloomquist, Zafer Asim Kaplancikli and Ahmet Ozdemir
DOI: 10.2174/1570180814666171002155548




Illicium verum Extract Exhibited Anti-inflammatory Action in Rodents

Volume:15   Issue: 6
Pp: 678-686
Shagufta Khan*, Huma Aslam Bhatti*, Ghulam Abbas, Muhammad Ali Versiani, Shaheen Faizi, Salman Khalid Ahmed, Saad Jawaid, Anita Naushir Akbar Ali, Rabia Jamy, Fatima Shahid and Ahsana Dar Farooq
DOI: 10.2174/1570180814666170915163236




Laser Modified Phenothiazines and Hydantoins: Photo-products Characterisation and Application on Animal Eyes Pseudo-tumours

Volume:15   Issue: 6
Pp: 687-697
Tatiana Tozar, Adriana Smarandache, Mihail Lucian Pascu*, Angela Staicu and Ruxandra Angela Pirvulescu
DOI: 10.2174/1570180814666170914115415