Letters in Drug Design & Discovery

Editor-in-Chief
K. Kuca
University of Hradec Kralove
Hradec Kralove
Czech Republic

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Volume:15   Issue: 4
Pp: 335-335
James David Adams
DOI: 10.2174/157018081504180312110402



Synthesis, Anti-Methicillin-resistant S. aureus (MRSA) Evaluation, Quantitative Structure-Activity Relationship and Molecular Modeling Studies of Some Novel Bis-indoles as Prospective MRSA Pyruvate Kinase Inhibitors

Volume:15   Issue: 4
Pp: 336-346
Mardia T. El Sayed*, Nermien M. Sabry, Nehal A. Hamdy, Andrey Voronkov, Ifedayo V. Ogungbe, Konstantin Balakin and Mohamed S. Abdel-Aziz
DOI: 10.2174/1570180815666171213144922



Anti-MRSA (Multidrug Resistant Staphylococcus aureus) Activity of 3-Substituted Coumarins

Volume:15   Issue: 4
Pp: 353-362
Uzma Salar, Khalid Mohammed Khan*, Humaira Muhammad, Muhammed Imran Fakhri, Sanaullah, Shahnaz Perveen and Muhammed Iqbal Choudhary
DOI: 10.2174/1570180814666170619121844



Synthesis and Anti-influenza Activity of Novel Thiadiazole, Oxadiazole and Triazole Based Scaffolds

Volume:15   Issue: 4
Pp: 363-374
Samar S. Tawfik, Abdelbasset A. Farahat*, Magda A.-A El-Sayed, Atif S. Tantawy, Ola Bagato and Mohamed A. Ali
DOI: 10.2174/1570180814666170512122832



Exploration of Some Thiazolidine-2,4-dione and 2-Oxoindoline Derivatives Incorporating 3,4,5-Trimethoxybenzyl Moiety as Novel Anticancer Agents

Volume:15   Issue: 4
Pp: 375-387
Le Cong Huan, Hai Pham-The, Huong Le-Thi-Thu, Tran Phuong Thao, Do Nguyet Que, Nguyen-Thu Trang, Phan Thi Phuong Dung, Minji Pyo, Sang-Bae Han, Nguyen Thi Thuan* and Nguyen-Hai Nam*
DOI: 10.2174/1570180814666170605122552



Design, Synthesis and Biological Evaluation of Some Novel Thiazole-2- Carboxamide Derivatives as Antitumor Agents

Volume:15   Issue: 4
Pp: 388-397
Haibo Wang*, Zhengjiang Cai, Shan Zheng, Huidan Ma, Haiming Lin and Xiaohe Zheng*
DOI: 10.2174/1570180814666170704143015



Fighting Against Alzheimer's Disease: Synthesis of New Pyrazoline and Benzothiazole Derivatives as New Acetylcholinesterase and MAO Inhibitors

Volume:15   Issue: 4
Pp: 414-427
Gulhan Turan-Zitouni*, Weiam Hussein, Begum Nurpelin Saglik, Merve Baysal and Zafer Asim Kaplancikli
DOI: 10.2174/1570180814666170704144917



Synthesis and Urease Inhibitory Activity of Some 5-Aminomethylene Barbituric/Thiobarbituric Acid Derivatives

Volume:15   Issue: 4
Pp: 428-436
Mehdi Asadi, Mohammad Mahdavi, Shabnam Mahernia, Zahra Rezaei, Maliheh Safavi, Mina Saeedi and Massoud Amanlou*
DOI: 10.2174/1570180814666170727142928