Letters in Drug Design & Discovery

Editor-in-Chief:

George Perry
University of Texas
San Antonio, TX
USA

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Volume:15   Issue:11
Pp: 1123-1123
Eng-Ang Ling
DOI: 10.2174/157018081511180925144148



Oxime K033-Reactivation Activity of Cholinesterases Inhibited by Various Nerve Agents and Organophosphorus Pesticides

Volume:15   Issue:11
Pp: 1124-1130
Kamil Kuca*, Kamil Musilek, Daniel Jun, Jaroslav Pejchal, Ondrej Krejcar, Marek Penhaker, Qinghua Wu, Raquel O. Lopes, Teodorico C. Ramalho, Tanos C.C. Franca, Eugenie Nepovimova and Ondrej Soukup
DOI: 10.2174/1570164615666180713112238



Design, Synthesis and Characterization of Novel Urolithin Derivatives as Cholinesterase Inhibitor Agents

Volume:15   Issue:11
Pp: 1131-1140
Maryam Norouzbahari, Emine V. Burgaz, Tugba Ercetin, Amirhossein Fallah, Alireza Foroumadi, Loghman Firoozpour, Mustafa F. Sahin, Mustafa Gazi and Hayrettin O. Gulcan*
DOI: 10.2174/1570180815666180115144608



Radioprotective Effect of Sinapic Acid Against Genotoxicity and Apoptosis Induced by Ionizing Radiation on Human Lymphocytes

Volume:15   Issue:11
Pp: 1147-1154
Fatemeh Alizadeh, Mohammad Asghari, Seyedeh Atekeh Torabizadeh, Najmeh Rahmanian, Arash Ghasemi and Seyed Jalal Hosseinimehr*
DOI: 10.2174/1570180815666180219163626



Inhibition of DNA Topoisomerases by a Series of Benzoxazoles and their Possible Metabolites

Volume:15   Issue:11
Pp: 1155-1162
Fatma Zilifdar*, Egemen Foto, Tugba Ertan-Bolelli, Ilkay Yildiz, Esin Aki-Yalcin and Nuran Diril
DOI: 10.2174/1570180815666180124143246



Averrhoa bilimbi L. leaf Aqueous Extract Modulates both Cardiac Contractility and Frequency in the Guinea-pig Atrium by the Activation of Muscarinic Receptors

Volume:15   Issue:11
Pp: 1163-1169
Anne Caroline Oliveira dos Santos, Diego Santos Souza, Thassio Ricardo Ribeiro Mesquita, Jose Evaldo Rodrigues de Menezes-Filho, Ana Paula Duarte Caldas, Americo Azevedo de Souza, Gilmara Beatriz Andrade da Silva, Evaleide Diniz de Oliveira, Leonardo Rodrigues dos Santos and Carla Maria Lins de Vasconcelos*
DOI: 10.2174/1570180815666180125150457



6-Methoxy-3,4-dihydronaphthalenone Chalcone-like Derivatives as Potent Tyrosinase Inhibitors and Radical Scavengers

Volume:15   Issue:11
Pp: 1170-1179
Sara Ranjbar, Abdolhossein Akbari, Najmeh Edraki, Mahsima Khoshneviszadeh, Hajar Hemmatian, Omidreza Firuzi and Mehdi Khoshneviszadeh*
DOI: 10.2174/1570180815666180219155027



Oral Bioavailability of Naturally Occurring Anticancer Phytomolecules

Volume:15   Issue:11
Pp: 1180-1188
Shilpa Sharma, Mansi Gupta, Ashish Sharma and Subhash M. Agarwal*
DOI: 10.2174/1570180815666180109161014



Design, Synthesis and Biological Evaluation of Novel Dihydropyrimidine- 2-Thione Derivatives as Potent Antimicrobial Agents: Experimental and Molecular Docking Approach

Volume:15   Issue:11
Pp: 1189-1201
Ehsan Ullah Mughal*, Amina Sadiq, Muhammad Hamayun, Muhammad Naveed Zafar, Nighat Fatima, Muhammad Arfat Yameen, Syed Aun Muhammad, Amara Mumtaz, Ishtiaq Ahmed and Tehseen Fatima
DOI: 10.2174/1570180815666180209151516



Synthesis, In Silico and Antifungal Studies of Novel Thiophene Analogues Containing Pyrazole Ring

Volume:15   Issue:11
Pp: 1202-1210
Helmi M. Al-Maqtari, Joazaizulfazli Jamalis*, Subhash Chander, Hasnah M. Sirat , Shivalingegowda Naveen, Neratur K. Lokanath, Siti P.M. Bohari, Deepak P. Bhagwat and Murugesan Sankaranarayanan
DOI: 10.2174/1570180815666180328144325



Molecular Docking and 3D-QSAR Studies on 7-azaindole Derivatives as Inhibitors of Trk A: A Strategic Design in Novel Anticancer Agents

Volume:15   Issue:11
Pp: 1211-1223
Adnane Aouidate*, Adib Ghaleb, Mounir Ghamali, Samir Chtita, Abdellah Ousaa, M`barek Choukrad, Abdelouahid Sbai, Mohammed Bouachrine and Tahar Lakhlifi
DOI: 10.2174/1570180815666171229151138



Synthetic Aspects and First-time Assessment of 2-amino-1,3-selenazoles Against Mycobacterium tuberculosis

Volume:15   Issue:11
Pp: 1224-1229
Victor Facchinetti, Marcus V.N. De Souza*, Ana C.S. Nery, Stephane L. Calixto, Juliana T. Granato, Elaine S. Coimbra, Maria C.S. Lourenco, Claudia R.B. Gomes and Thatyana R.A. Vasconcelos
DOI: 10.2174/1570180815666180209153925



Synthesis, Characterization and Evaluation of Gemfibrozil-Stilbene Hybrid as Antioxidant Agent

Volume:15   Issue:11
Pp: 1230-1238
Rosa Amoroso, Lidia Leporini, Ivana Cacciatore, Lisa Marinelli, Alessandra Ammazzalorso, Isabella Bruno, Barbara De Filippis, Marialuigia Fantacuzzi, Cristina Maccallini, Luigi Menghini, Antonio Di Stefano and Letizia Giampietro*
DOI: 10.2174/1570180815666180321163246