Letters in Drug Design & Discovery

Editor-in-Chief:

George Perry
University of Texas
San Antonio, TX
USA

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Volume:14   Issue:4
Pp: 373-373
Romano Silvestri
DOI: 10.2174/157018081404170223193954



Quinoline Derivatives as Novel Depigmenting and Antioxidant Agents

Volume:14   Issue:4
Pp: 374-379
Rebeca Mol Lima, Kauana Cristina de Souza, Jordana de Abreu Lazzarini, Isabela O. Souza, Adilson David da Silva and Nadia Rezende Barbosa Raposo
DOI: 10.2174/1570180813666160930164926



Synthesis and Antioxidant Activity of Indole Derivatives Containing 4-Substituted Piperazine Moieties

Volume:14   Issue:4
Pp: 380-386
Tunca Gul Altuntas, Nilüfer Yılmaz, Tulay Coban and Sureyya Olgen
DOI: 10.2174/1570180813666161020165623



Synthesis, Antiproliferative, and Antiangiogenic Activities of Benzochromene and Benzoquinoline Derivatives on Prostate Cancer in vitro

Volume:14   Issue:4
Pp: 398-413
Gricelda Mata, Juan Rodrigues, Neira Gamboa, Katiuska Charris, Gricela Lobo, Melina Monasterios, Milagros Avendano, Michael Lein, Klaus Jung, Claudia Abramjuk, Bianca Nitzsche, Michael Hopfner and Jaime Charris
DOI: 10.2174/1570180814666161118163844



3D-QSAR and Molecular Docking Studies of Pyrazole Derivatives as Inhibitors of Enoyl Acyl Carrier Protein Reductase from Mycobacterium tuberculosis

Volume:14   Issue:4
Pp: 414-433
Sheshagiri R. Dixit, Shrinivas D. Joshi, V. H. Kulkarni and Tejraj M. Aminabhavi
DOI: 10.2174/1570180814666161107155459



Synthesis, Molecular Docking and Pharmacological Study of Pyrimidothiadiazinones and its bis-derivatives

Volume:14   Issue:4
Pp: 434-443
Sobhi M. Gomha, Ikhlass M. Abbas, Mohamed A. A. Elneairy, Mahmoud M. Elaasser and Bazada K. A. Mabrouk
DOI: 10.2174/1570180813666160815125409



Structure-Based Hybridization, Conventional and Microwave Irradiated Synthesis, Biological Evaluation and Molecular Docking Studies of New Compounds Derived from Thiomorpholin

Volume:14   Issue:4
Pp: 444-463
Serpil Demirci, Fatma Aksakal, Nesrin Colak, Serdar Ulker, Ahmet Demirbas and Neslihan Demirbas
DOI: 10.2174/1570180813666161024165613



Improved Anti-inflammatory Activity and Potential Cytoprotective Properties of Tolfenamic Acid, Naproxen and Indomethacin Derivatives

Volume:14   Issue:4
Pp: 464-475
Panagiotis Theodosis-Nobelos, Theodora C. Politou, Chrysoula Athanasekou and Eleni A. Rekka
DOI: 10.2174/1570180813666160831143112



Chronobiotic Hormone Melatonin: Comparative in vitro Release Studies from Matrix Tablets and Liposomal Formulations

Volume:14   Issue:4
Pp: 476-480
Androniki Zampakola, Angeliki Siamidi, Natassa Pippa, Costas Demetzos and Marilena Vlachou
DOI: 10.2174/1570180813666161006162246



Caffeic Acid Phenethyl Ester Restores Adipocyte Gene Profile Expression Following Lipopolysaccharide Treatment

Volume:14   Issue:4
Pp: 481-487
Ignazio Barbagallo, Giovanni Li Volti, Valeria Sorrenti, Claudia Di Giacomo, Rosaria Acquaviva, Marco Raffaele, Fabio Galvano and Luca Vanella
DOI: 10.2174/1570180813666160901124707



Sequential Therapy For Helicobacter pylori in Elderly Patients: Effectiveness, Safety and Predictors of Success

Volume:14   Issue:4
Pp: 500-505
Giuseppe Losurdo, Andrea Iannone, Floriana Giorgio, Michele Barone, Mariabeatrice Principi, Enzo Ierardi and Alfredo Di Leo
DOI: 10.2174/1570180813666160922113541