Letters in Drug Design & Discovery

Editor-in-Chief
K. Kuca
University of Hradec Kralove
Hradec Kralove
Czech Republic

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Volume:14   Issue: 11
Pp: 1227-1227
Eliezer J. Barreiro
DOI: 10.2174/157018081411171003112446



2D, 3D, G-QSAR and Docking Studies of Thiazolyl-pyrazoline Analogues as Potent (Epidermal Growth Factor Receptor-tyrosine Kinase) EGFR-TK Inhibitors

Volume:14   Issue: 11
Pp: 1228-1238
Ghodgaonkar Sunayana*, Bhandari Shashikant and Waghulde Sandeep
DOI: 10.2174/1570180814666170518171236




Synthesis, Docking and Evaluation of Phenylacetic Acid and Trifluoro-methylphenyl Substituted Benzamide Derivatives as Potential PPARδ Agonists

Volume:14   Issue: 11
Pp: 1239-1251
Ajmer Singh Grewal, Viney Lather*, Deepti Pandita and Garima Bhayana
DOI: 10.2174/1570180814666170327164443




Molecular Docking Studies of Novel Thiosemicarbazone-based Indoles as Potential PI3Kα Inhibitors

Volume:14   Issue: 11
Pp: 1252-1258
Dima A. Sabbah* and Kamal Sweidan
DOI: 10.2174/1570180814666170619112647




Synthesis and Structure-activity Relationships of Chalcone Derivatives as Inhibitors of Ovarian Cancer Cell Growth

Volume:14   Issue: 11
Pp: 1259-1266
Zachary D. Tucker, Francis J. Barrios and Amanda J. Krzysiak*
DOI: 10.2174/1570180814666170505120258




Molecular Docking and In Silico ADMET Study Reveals Flavonoids as a Potential Inhibitor of Aromatase

Volume:14   Issue: 11
Pp: 1267-1276
Umang Shah*, Samir Patel, Mehul Patel and Jagat Upadhayay
DOI: 10.2174/1570180814666170327161908




Molecular Simulation and Activity Studies of Oxametacin as an HDAC Inhibitor

Volume:14   Issue: 11
Pp: 1277-1282
Fanbo Jing, Lei Zhang*, Yepeng Luan and Jiang Bian
DOI: 10.2174/1570180814666170505123930




The Antiviral Effects of Harmine Against BoHV-1 Infection In Vitro

Volume:14   Issue: 11
Pp: 1303-1307
Xinyi Jiang, Jie Zou, Yuncheng Zhuang, Weifeng Yuan, Liqian Zhu* and Guoqiang Zhu*
DOI: 10.2174/1570180814666170425155554




New Cyclohexylamine-dithiocarbamate Derivatives as Potential Anti-microbial Agents

Volume:14   Issue: 11
Pp: 1308-1315
Leyla Yurttas*, Betul Kaya , Meral Yilmaz Cankilic and Serkan Levent
DOI: 10.2174/1570180814666170412121402




Synthesis and Antimicrobial Activity of Some Novel Substituted 3-(Thiophen-2-yl)pyrazole-based Heterocycles

Volume:14   Issue: 11
Pp: 1316-1323
Bakr F. Abdel-Wahab*, Abdelbasset A. Farahat, Ghada E. A. Awad and Gamal A. El-Hiti*
DOI: 10.2174/1570180814666170327162447




Novel Thiazole Carboxylic Acid Derivatives Possessing a “Zinc Binding Feature” as Potential Human Glyoxalase-I Inhibitors

Volume:14   Issue: 11
Pp: 1324-1334
Qosay A. Al-Balasa*, Mohammad A. Hassana, Ghazi A. Al Jabala, Nizar A. Al-Shar, Ammar M. Almaaytahb and Tamam El-Elimata
DOI: 10.2174/1570180814666170306120954




Synthesis and Antiproliferative Activity of 3-aza Steroids as 5α-reductase Inhibitors

Volume:14   Issue: 11
Pp: 1335-1346
Milanpreet Kaur, Richa Dhingra, T. R. Bhardwaj and Neelima Dhingra*
DOI: 10.2174/1570180814666170505122503