Letters in Drug Design & Discovery

Editor-in-Chief:

George Perry
University of Texas
San Antonio, TX
USA

Back

Become EABM
Become Reviewer

Design, Synthesis and ex vivo Study of the Vasorelaxant Activity Induced by Isosteric Derivatives of Dihydropyridines (NH→O)

Volume:13   Issue:5
Pp: 353-359
Priscila Rendón-Vallejo, Samuel Estrada-Soto, Miguel A. Vázquez, Fernando Hernández- Borja, Rafael Villalobos-Molina and Maximiliano Ibarra-Barajas
DOI: 10.2174/1570180812666151003002501

Flexibility in the Molecular Design of Acetylcholinesterase Reactivators: Probing Representative Conformations by Chemometric Techniques and Docking/QM Calculations

Volume:13   Issue:5
Pp: 360-371
Willian E.A. de Lima, Ander F. Pereira, Alexandre A. de Castro, Elaine F.F. da Cunha and Teodorico C. Ramalho
DOI: 10.2174/1570180812666150918191550

TRISOXIME – a Bulky Trisquaternary Reactivator of Acetylcholinesterase

Volume:13   Issue:5
Pp: 372-375
Kamil Kuca, Kamil Musilek and Daniel Jun
DOI: 10.2174/1570180812666150923235240

CoMFA/CoMSIA and Molecular Docking Studies of Novel Matrix Metalloproteinase- 2 Inhibitors Based on L-tyrosine Scaffold

Volume:13   Issue:5
Pp: 376-386
Jun-Zhang, Xue-Jiao Wang, Zhen-Ke Dong, Shu-Qing Wang, Wei-Ren Xu, Jing-Wei Fu, Xian- Chao Cheng and Run-Ling Wang
DOI: 10.2174/1570180812666150923235104

Synthesis, Neuro-protection and Anti-cancer Activities of Simple Isatin Mannich and Schiff Bases

Volume:13   Issue:5
Pp: 395-400
Gang Chen, Yang Ning, Wei Zhao, Yanqiu Zhang, Yu Zhang, Xiaojiang Hao, Ye Wang and Shuzhen Mu
DOI: 10.2174/1570180812666150907203342

Modified Hummel-Dreyer Method and Molecular Modeling Studies Identified Nicotinic Acid Analogues as Carbonic Anhydrase III Ligands

Volume:13   Issue:5
Pp: 401-410
Nada Jarrar, Muhammed Alzweiri, Yusuf Al-Hiari, Shrouq Farah and Mohammad A. Khanfar
DOI: 10.2174/1570180812666150821002900

In vitro Study of Furazano[3,4-b]quinoxaline 1-Oxides as Potential ΝΟ Releasing Agents

Volume:13   Issue:5
Pp: 418-421
Kosmas I. Stoitsis, Petros Gkizis, Emmanouella Basgiouraki, John K. Gallos and Dimitra Hadjipavlou-Litina
DOI: 10.2174/1570180812666150923235828

Design, Synthesis and Mode of Action of Some New 2-(4'-aminophenyl) benzothiazole Derivatives as Potent Antimicrobial Agents

Volume:13   Issue:5
Pp: 429-437
Meenakshi Singh, Sudhir Kumar Singh, Mayank Gangwar, Satheeshkumar Sellamuthu, Gopal Nath and Sushil K. Singh
DOI: 10.2174/1570180812666150821003220

Accumulation Effects of Salicylic acid Saccharide Carboxylate on the Alkaloids in Catharanthus roseus Cells

Volume:13   Issue:5
Pp: 438-440
Er-Bing Yang, Yong Wang, Hong-Jun Zang, Zheng-Ming Li and Xing-Hai Liu
DOI: 10.2174/1570180812666150818235025

Despite an Extensive Sequence Analysis Identification of Functional Candidates Amongst Hypothetical Proteins of Neisseria gonorrhoeae

Volume:13   Issue:5
Pp: 451-464
Kundan Kumar, Amresh Prakash, Asimul Islam, Faizan Ahmad and Md. Imtaiyaz Hassan
DOI: 10.2174/1570180812666150901223055

Sunscreening and Photosensitizing Properties of Coumarins and their Derivatives

Volume:13   Issue:5
Pp: 465-474
Kinga Kasperkiewicz, Anna Erkiert-Polguj and Elzbieta Budzisz
DOI: 10.2174/1570180812666150901222106