Letters in Drug Design & Discovery

Editor-in-Chief
K. Kuca
University of Hradec Kralove
Hradec Kralove
Czech Republic

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Volume:12   Issue: 5
Pp: 343-343
Mihail Lucian Pascu
DOI: 10.2174/157018081205150324101302

Discovery of Novel HDAC Inhibitors by Structure-based Optimization of Cinnamic Hydroxamic Scaffold

Volume:12   Issue: 5
Pp: 344-350
Chengqing Ning, Wenyuan Huang, Wen Wu, Cheng Lu, Yujun He, Lei Yao, Lifei Liu, Xiaohe Zhen, Xiaoyu Liu and Niefang Yu
DOI: 10.2174/1570180811666141024004832

Development of Structure Activity Correlation Model on Azetidin-2-ones as Tubulin Polymerization Inhibitors

Volume:12   Issue: 5
Pp: 351-365
Vijay Kumar Patel, Kavibhushan Singh Chouhan, Avineesh Singh, Deepak Kumar Jain, Ravichandran Veerasamy, Pradeep Kumar. Singour, Rajesh Singh Pawar and Harish Rajak
DOI: 10.2174/1570180811666141010000110

Synthesis and Anticancer Activity of 7,8-dihydroxy-4-arylcoumarins

Volume:12   Issue: 5
Pp: 366-373
Jianrui Wu, Ting Peng, Fang Chen, Yixin Leng, Linjiang Tong, Mengyuan Li, Rong Qu, Hua Xie, Jian Ding and Wenhu Duan
DOI: 10.2174/1570180812666141111235026

Hybrid Pharmacophore Design and Synthesis of Naphthalimide– Benzimidazole Conjugates as Potential Anticancer Agents

Volume:12   Issue: 5
Pp: 374-384
Ahmed Kamal, Pogula Praveen Kumar, Mohammed Naseer Ahmed Khan, Bobburi Naga Sheshadri and Naga Sheshadri
DOI: 10.2174/1570180811666140915221955

Promising Anticancer Drug Candidates Based on the 7-methoxychromone Scaffold: Synthesis and Evaluation of Antiproliferative Activity

Volume:12   Issue: 5
Pp: 385-392
Hoang Le Tuan Anh, Nguyen Thi Cuc, Pham Hai Yen, Nguyen Xuan Nhiem, Bui Huu Tai, Do Thi Thao, Nguyen Hoai Nam, Chau Van Minh, Phan Van Kiem and Young Ho Kim
DOI: 10.2174/1570180812666141111235539

Design, Synthesis and Biological Evaluation of Novel Fluorinated Heterocyclic Hybrid Molecules Based on Triazole & Quinoxaline Scaffolds Lead to Highly Potent Antimalarials and Antibacterials

Volume:12   Issue: 5
Pp: 393-407
Adimulam Chandra Shekhar, Boddupally Pedda Venkat Lingaiah, Pamulaparthy Shanthan Rao, Banda Narsaiah, Aparna Devi Allanki and Puran Singh Sijwali
DOI: 10.2174/1570180812666141111235301

Synthesis of Derivatives of Artesunate α-Aminophosphonate and Their Antimicrobial Activities

Volume:12   Issue: 5
Pp: 408-416
Sheng He, Xilin Ouyang, Xiaochao Huang, Weisong Hu, Weilong Dai, Xiaoyan Tian, Yingming Pan, Shiwen Huang and Hengshan Wang
DOI: 10.2174/1570180812666141125004502

Synthesis and Preliminary Biological Evaluation of New Heterocyclic Carboxamide Models

Volume:12   Issue: 5
Pp: 417-429
Kamal Sweidan, Jorn Engelmann, Walid Abu Rayyan, Dima Sabbah, Musa Abu Zarga, Dima Sabbah, Tariq Al-Qirim, Yusuf Al-Hiari, Ghassan Abu Sheikha and Ghassan Shattat
DOI: 10.2174/1570180812666141201222527