Letters in Drug Design & Discovery


George Perry
University of Texas
San Antonio, TX


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Volume:10   Issue:6
Pp: i-iv

DOI: 10.2174/1570180811310060001

Synthesis of New Compounds Combining Adamantanamine and Monoterpene Fragments and their Antiviral Activity Against Influenza Virus A(H1N1)pdm09

Volume:10   Issue:6
Pp: 477-485
George V. Teplov, Evgeny V. Suslov, Vladimir V. Zarubaev, Anna A. Shtro, Liubov A. Karpinskaya, Artem D. Rogachev, Dina V. Korchagina, Konstantin P. Volcho, Nariman F. Salakhutdinov and Oleg I. Kiselev
DOI: 10.2174/1570180811310060002

Synthesis and Antimicrobial Evaluation of Some 2,5-Disubstituted Benzimidazole Derivatives

Volume:10   Issue:6
Pp: 486-491
Leyla Yurttas, Yusuf Ozkay, Hulya Karaca, Yagmur Tunali and Zafer Asim Kaplancıkli
DOI: 10.2174/1570180811310060003

Diversity in Antibacterial Activity of Thiosemicarbazides Derived from 3-Chlorobenzhydrazide

Volume:10   Issue:6
Pp: 492-496
Tomasz Plech, Monika Wujec, Urszula Kosikowska and Anna Malm
DOI: 10.2174/1570180811310060004

Synthesis of Novel 3-Chloropyridin-2-yl-Pyrazole Derivatives and their Insecticidal, Fungicidal Activities and QSAR Study

Volume:10   Issue:6
Pp: 497-506
Ji-Feng Zhang, Chen Liu, Yi Ma, Bao-Lei Wang, Li-Xia Xiong, Shu-Jing Yu and Zheng-Ming Li
DOI: 10.2174/1570180811310060005

Synthesis of Some New 3(2H)-Pyridazinone Derivatives and Evaluation of their Analgesic-anti-inflammatory and Antimicrobial Activities

Volume:10   Issue:6
Pp: 507-514
Murat Sukuroglu, Cem Yamali, Didem Tiryaki, Fatma Kaynak Onurdag, Esra Akkol and Deniz Songul Dogruer
DOI: 10.2174/1570180811310060006

Discovery and Study of the Binding Epitopes of Novel Urease Inhibitors by STD-NMR Spectroscopy and Biochemical Analyses

Volume:10   Issue:6
Pp: 515-521
Atia-tul- Wahab, Ajmal Khan, Bishnu P. Marasini, M. Arif Lodhi, Atta-ur- Rahman and M. Iqbal Choudhary
DOI: 10.2174/1570180811310060007

Design, Synthesis and Evaluation of Arylidene Pyrrolo and Pyrido Fused Quinazolones as Antimicrobial Agents

Volume:10   Issue:6
Pp: 522-528
Kunal Nepali, Ritu Ojha, Aninder Singh, Abhishek Budhiraja, Preet Mohinder Singh Bedi and Kanaya Lal Dhar
DOI: 10.2174/1570180811310060008

Inhibitory Effects of Substituted Cinnamic Acid Esters on Mushroom Tyrosinase

Volume:10   Issue:6
Pp: 529-534
Zhenghua Zhang, Jinbing Liu, Fengyan Wu and Liangzhong Zhao
DOI: 10.2174/1570180811310060009

Improved Pharmacokinetic Profile and Anti-Inflammatory Property of a Novel Curcumin Derivative, A50

Volume:10   Issue:6
Pp: 535-542
Xiangjian Chen, Luqing Ren, Xiuhua Zhang, Lu Guo, Jianmin Zhou, Guang Liang and Yi Wang
DOI: 10.2174/1570180811310060010

Synthesis and Evaluation of the Anticonvulsant Activity of 5-alkylthio-4- phenyl-2,4-dihydro-3H-1,2,4-triazol-3-one Derivatives

Volume:10   Issue:6
Pp: 543-549
Yan Zheng, Xian-Qing Deng, Bing Shu, Shi-Ben Wang, Xu Cao and Zhe-Shan Quan
DOI: 10.2174/1570180811310060011

Curcumin Activates Erythrocyte Membrane Acetylcholinesterase

Volume:10   Issue:6
Pp: 550-556
Prabhakar Singh and Syed Ibrahim Rizvi
DOI: 10.2174/1570180811310060012