Letters in Drug Design & Discovery

Editor-in-Chief:

George Perry
University of Texas
San Antonio, TX
USA

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Graphical Abstracts promotion: free to download

Volume:10   Issue:1
Pp: i-iv

DOI: 10.2174/157018081130901000i



Editorial free to download

Volume:10   Issue:1
Pp: 1-1
Atta-ur-Rahman
DOI: 10.2174/1570180811309010001

Search for Molecular Basis of Antifungal Activity of Thiosemicarbazide Derivatives: A Combined in vitro Antifungal and Enzymatic Studies with in Silico Docking promotion: free to download

Volume:10   Issue:1
Pp: 2-10
Agata Siwek, Pawel Staczek, Aleksandra Strzelczyk and Joanna Stefanska
DOI: 10.2174/1570180811309010002

Boronic Acid Based Inhibitors of Autotaxin: Understanding their Biological Role in Terms of Quantitative Structure Activity Relationships (QSAR) promotion: free to download

Volume:10   Issue:1
Pp: 11-18
Sotirios Katsamakas and Dimitra Hadjipavlou-Litina
DOI: 10.2174/1570180811309010011

Synthesis and Biological Study of Novel Indole-3-Imine-2-on Derivatives as Src Kinase and Glutathione S-Transferase Inhibitors promotion: free to download

Volume:10   Issue:1
Pp: 19-26
Z. Kilic Kurt, D. Aydin, Y. G. Isgor, B. S. Isgor and S. Olgen
DOI: 10.2174/1570180811309010019

Synthesis and Anti-HIV Evaluation of Novel 1,2,4-triazole Derivatives as Potential Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors promotion: free to download

Volume:10   Issue:1
Pp: 27-34
Zhenyu Li, Yuan Cao, Peng Zhan, Christophe Pannecouque, Jan Balzarini, Erik De Clercq and Xinyong Liu
DOI: 10.2174/1570180811309010027

Synthesis and Evaluation of Anticonvulsant Activity of Some N-[(4-Chlor- 2-methylphenoxy)ethyl]- and N-[(4-Chlor-2-methylphenoxy)acetyl]aminoalkanols promotion: free to download

Volume:10   Issue:1
Pp: 35-43
Anna M. Waszkielewicz, Edward Szneler, Marek Cegla and Henryk Marona
DOI: 10.2174/1570180811309010035

Synthesis and Antimicrobial Activity of some Amide Derivatives Bearing Thiazole, Benzhydryl and Piperidine Moieties promotion: free to download

Volume:10   Issue:1
Pp: 44-48
Ahmet Ozdemir
DOI: 10.2174/1570180811309010044

Protein Interaction Networks in Metallo Proteins and Docking Approaches of Metallic Compounds with TIMP and MMP in Control of MAPK Pathway promotion: free to download

Volume:10   Issue:1
Pp: 49-55
Kaladhar Svgk Dowluru, Potladurthi Chandra Sai, Padmanabhuni Venkata Nageswara Rao, Amajala Krishna chaitanya, Duddukuri Govinda Rao, Vadlapudi Varahala Rao, Potladurthi Suresh, Erva Rajeswara Reddy, Sudabattula Vijaya kumar, Divyakolu Vinod Kumar and Gajjala Bhaskar Reddy
DOI: 10.2174/1570180811309010049

Evaluation of In-Vitro Multidrug Resistance Reversal Activities of HZ08 analogues with Improved Soluble Property promotion: free to download

Volume:10   Issue:1
Pp: 56-60
Xiaobu Lan, Haiyan Lin, Chunlei Tang, Xiaoyun Zhu, Hai Qian, Wenlong Huang and Yunman Li
DOI: 10.2174/1570180811309010056

Synthesis and Antiproliferative Evaluation of Hybrids of Indolin-2-one and Quinazoline-4(3H)-one Linked via Imine Bond promotion: free to download

Volume:10   Issue:1
Pp: 61-66
Wei-Yao Wu, Sheng-Li Cao, Bei-Bei Mao, Ji Liao, Zhong-Feng Li, Hao-Bin Song and Xingzhi Xu
DOI: 10.2174/1570180811309010061

Identification of Leads from Marine Seaweeds against Human β-tubulin promotion: free to download

Volume:10   Issue:1
Pp: 67-74
Selvaa Kumar C, Nikhil Gadewal and Sudheer M.M. Mohammed
DOI: 10.2174/1570180811309010067

Design, Synthesis and Evaluation of Novel 2-piperidinyl Quinoline Chalcones/ Amines as Potential Antidepressant Agents promotion: free to download

Volume:10   Issue:1
Pp: 75-85
Obaid Afzal, Sandhya Bawa, Suresh Kumar, Rajiv Kumar and Md Quamrul Hassan
DOI: 10.2174/1570180811309010075

Synthesis, Characterization, Antimicrobial Activity of Novel N-Substituted β-Hydroxy Amines and βHydroxy Ethers Contained Chiral Benzoxazine Fluoroquinolones promotion: free to download

Volume:10   Issue:1
Pp: 86-93
B. Guruswamy and R. Arul
DOI: 10.2174/1570180811309010086