Letters in Drug Design & Discovery

Editor-in-Chief
K. Kuca
University of Hradec Kralove
Hradec Kralove
Czech Republic

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Volume 16 - Issue 12



Meet Our Associate Editor promotion: free to download

Volume: 16   Issue: 12
Pp: 1303-1304
Bimal Krishna Banik
DOI: 10.2174/157018081612191108153022



Effects of Acute and Chronic Treatment of Novel Psychotropic Drug, 8- (Trifluoromethyl)-1, 2, 3, 4, 5-benzopentathiepin-6-amine Hydrochloride (TC-2153), on the Behavior of Zebrafish (Danio Rerio): A Comparison with Fluoxetine

Volume: 16   Issue: 12
Pp: 1321-1328
Alexander Kulikov, Nadezhda Sinyakova, Elizabeth Kulikova, Tatyana Khomenko, Nariman Salakhutdinov, Victor Kulikov and Konstantin Volcho*
DOI: 10.2174/1570180816666190221162952



Biology-oriented Drug Synthesis (BIODS), Structural Characterization and Bioactivities of Novel Albendazole Derivatives

Volume: 16   Issue: 12
Pp: 1329-1338
Momin Khan*, Shahid Khan, Uzma Salar, Khalid Mohammed Khan, Gauhar Rehman, Naeem Gul and Iltaf Khan
DOI: 10.2174/1570180816666190221163641



Baicalin-induced Cytotoxicity and Apoptosis in Multidrug-resistant MC3/5FU Mucoepidermoid Carcinoma Cell Line

Volume: 16   Issue: 12
Pp: 1339-1347
Xiaofang Xu, Qihong Li, Kaitao Yu*, Ghulam Murtaza* and Bin Liu*
DOI: 10.2174/157018081210151012121717



Design, Synthesis and Bioactivity of Core 1 O-glycan and its Derivative on Human Gut Microbiota

Volume: 16   Issue: 12
Pp: 1348-1353
Huanhuan Qu*, Baixue Li, Jingyi Yang, Huaiwen Liang, Meixia Li and Kan Ding*
DOI: 10.2174/1570180816666181218143207



Anticancer Potential of Pulicaria crispa Extract on Human Breast Cancer MDA-MB-231 Cells

Volume: 16   Issue: 12
Pp: 1354-1359
Ibrahim Omar Barnawi and Imran Ali*
DOI: 10.2174/1570180816666190712110224



Synthesis and Antimicrobial Activity of Adamantyl Substituted Pyridoxine Derivatives

Volume: 16   Issue: 12
Pp: 1360-1369
Rail Khaziev, Nikita Shtyrlin, Roman Pavelyev, Raushan Nigmatullin, Raylya Gabbasova, Denis Grishaev, Anna Shtro, Anastasia Galochkina , Yulia Nikolaeva , Tatiana Vinogradova , Olga Manicheva, Marine Dogonadze, Oleg Gnezdilov , Evgenii Sokolovich, Petr Yablonskiy, Konstantin Balakin and Yurii Shtyrlin*
DOI: 10.2174/1570180816666190911150705



The Antiviral Effects of Sodium Phenylbutyrate Against BoHV-1 Infection In Vitro

Volume: 16   Issue: 12
Pp: 1370-1377
Xinye Chen, Guoqiang Zhu* and Liqian Zhu*
DOI: 10.2174/1570180816666190222155958



Design, Synthesis and Biological Evaluation of Camptothecin Conjugated with NSAIDs as Novel Dual-actin Antitumor Agents

Volume: 16   Issue: 12
Pp: 1378-1386
Xingchen Cai, Weiwei Huang, Yi Huang, Lihua Xia, Miao Liu, Mengke Wang, Wenchao Wang and Qingyong Li*
DOI: 10.2174/1570180816666190221103257



Challenges in the Discovery and Optimization of mGlu2/4 Heterodimer Positive Allosteric Modulators open access plus

Volume: 16   Issue: 12
Pp: 1387-1394
Mark Gallant Fulton, Matthew Thomas Loch, Caroline Anne Cuoco, Alice Lambert Rodriguez, Emily Days, Paige Newton Vinson, Krystian Andrezej Kozek, Charles David Weaver, Anna Louise Blobaum, Peter Jeffrey Conn, Colleen Marie Niswender* and Craig William Lindsley*
DOI: 10.2174/1570180815666181017131349



Acknowledgements to Reviewers promotion: free to download

Volume: 16   Issue: 12
Pp: 1395-1396

DOI: 10.2174/157018081612191108153118