Letters in Drug Design & Discovery

Editor-in-Chief:

George Perry
University of Texas
San Antonio, TX
USA

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Volume 16 - Issue 5



Opportunities and Challenges in the Anticandidal Drug Discovery and Development promotion: free to download

Volume: 16   Issue: 5
Pp: 477-477
Mohammad Abid
DOI: 10.2174/157018081605190415121529



Potential of Nanoparticles in Combating Candida Infections

Volume: 16   Issue: 5
Pp: 478-491
Faizan Abul Qais, Mohd Sajjad Ahmad Khan, Iqbal Ahmad* and Abdullah Safar Althubiani
DOI: 10.2174/1570180815666181015145224



Recent Advances in Azole Based Scaffolds as Anticandidal Agents

Volume: 16   Issue: 5
Pp: 492-501
Prabhuodeyara Math Gurubasavaraj* and Jasmith Shivayya Charantimath
DOI: 10.2174/1570180815666180917125916



Phenolic Composition and Antifungal Effect of Costus cf. arabicus L Against Yeast of the Candida Genus

Volume: 16   Issue: 5
Pp: 502-511
Antonia Thassya Lucas Dos Santos, Antonio Júdson Targino Machado, Maria Audilene De Freitas, Irwin Rose Alencar De Menezes, Henrique Douglas Melo Coutinho, Francisco Assis Bezerra Da Cunha, Djair Dos Santos De Lima E Souza*, Aline Augusti Boligon, Adeliana Silva De Oliveira, Andressa De Alencar Silva and Maria Flaviana Bezerra Morais-Braga*
DOI: 10.2174/1570180815666180827122526



Synthesis and Anticancer Activity of New Hydrazide-hydrazones and Their Pd(II) Complexes

Volume: 16   Issue: 5
Pp: 522-532
Bedia Kocyigit-Kaymakcioglu*, Senem Sinem Yazici, Fatih Tok, Miriş Dikmen, Selin Engür, Emine Elçin Oruc-Emre and Aysegul Iyidogan
DOI: 10.2174/1570180815666180816124102



Design, Synthesis and Antitumor Activity of Quinazoline Derivatives Bearing 2,3-Dihydro-indole or 1,2,3,4-Tetrahydroquinoline

Volume: 16   Issue: 5
Pp: 533-546
Yiqiang OuYang, Bingbing Zhao, Xiuying Chen, Caolin Wang, Hong Zhang, Shuang Jia, Wufu Zhu* and Pengwu Zheng*
DOI: 10.2174/1570180815666180801121220



Novel Tri-substituted Thiazoles Bearing Piperazine Ring: Synthesis and Evaluation of their Anticancer Activity

Volume: 16   Issue: 5
Pp: 547-555
Asaf Evrim Evren*, Leyla Yurttaş, Busra Eksellı and Gulsen Akalın-Cıftcı
DOI: 10.2174/1570180815666180731122118



Cytotoxicity of Sodium Arsenite-loaded Anti-HER2 Immunoliposomes Against HER2-expressing Human Breast Cancer Cell Lines

Volume: 16   Issue: 5
Pp: 556-562
Moslem Afrakhteh, Alireza Kheirollah, Aminollah Pourshohod, Mohammad Ali Ghaffari, Mostafa Jamalan* and Majid Zeinali*
DOI: 10.2174/1570180815666180803120409



A Comparative Study of the Cytotoxic and Pro-apoptotic Properties of Nepeta binaloudensis

Volume: 16   Issue: 5
Pp: 563-569
Seyed Ahmad Emami, Hadi Al-Najjar, Javad Asili, Maryam Sadat Habibi, Amirhossein Sahebkar and Zahra Tayarani-Najaran*
DOI: 10.2174/1570180815666180918162805



In Silico Design of New B-Raf Kinase Type-II Inhibitors Through Combined Molecular Modeling Studies

Volume: 16   Issue: 5
Pp: 570-583
Weineng Zhou, Shuai Lu, Yanmin Zhang, Lingfeng Yin, Lu Zhu, Junnan Zhao, Tao Lu, Yadong Chen* and Haichun Liu*
DOI: 10.2174/1570180815666180816121628



Molecular Dynamics and Inhibition of MERS CoV Papain-like Protease by Small Molecule Imidazole and Aminopurine Derivatives

Volume: 16   Issue: 5
Pp: 584-591
Mahmoud Kandeel*, Abdallah Altaher and Mohamed Alnazawi
DOI: 10.2174/1570180815666180918161922



The Impacts of Some Sedative Drugs on α -Glycosidase, Acetylcholinesterase and Butyrylcholinesterase Enzymes-potential Drugs for Some Metabolic Diseases

Volume: 16   Issue: 5
Pp: 592-596
Ruya Kaya, Parham Taslimi*, Muhammet Emin Naldan and İlhami Gulçin
DOI: 10.2174/1570180815666180924110023



The Development of Tyrosyl-DNA Phosphodyesterase 1 (TDP1) Inhibitors Based on the Amines Combining Aromatic/Heteroaromatic and Monoterpenoid Moieties

Volume: 16   Issue: 5
Pp: 597-605
Evgenii Mozhaitsev, Evgenii Suslov*, Yuliya Demidova, Dina Korchagina, Konstantin Volcho, Alexandra Zakharenko, Inna Vasil'eva, Maksim Kupryushkin, Arina Chepanova, Daniel Moscoh Ayine-Tora, Jóhannes Reynisson, Nariman Salakhutdinov and Olga Lavrik
DOI: 10.2174/1570180816666181220121042