Letters in Drug Design & Discovery

Editor-in-Chief
K. Kuca
University of Hradec Kralove
Hradec Kralove
Czech Republic

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Most Accessed Articles

Design, Synthesis and Anti Colon Cancer Activity Evaluation of Phosphorylated Derivatives of Lamivudine (3TC) promotion: free to download

Volume: 8   Issue: 1
Pp: 59-64
Valasani Koteswara Rao, Sanapalli S. Reddy, Balam S. Krishna, Cirandur S. Reddy, Nimmanapalli P. Reddy, Tamatam C.M. Reddy, Chamarthi N. Raju and S. K. Ghosh
DOI: 10.2174/157018011793663921

Synthesis and Antimicrobial Activity of Adamantyl Substituted Pyridoxine Derivatives

Volume: 16   Issue: 12
Pp: 1360-1369
Rail Khaziev, Nikita Shtyrlin, Roman Pavelyev, Raushan Nigmatullin, Raylya Gabbasova, Denis Grishaev, Anna Shtro, Anastasia Galochkina , Yulia Nikolaeva , Tatiana Vinogradova , Olga Manicheva, Marine Dogonadze, Oleg Gnezdilov , Evgenii Sokolovich, Petr Yablonskiy, Konstantin Balakin and Yurii Shtyrlin*
DOI: 10.2174/1570180816666190911150705

Synthesis of Phenyl- and Pyridyl-substituted Benzyloxybenzaldehydes by Suzuki-Miyaura Coupling Reactions open access plus

Volume: 16   Issue: 11
Pp: 1248-1257
Hedvig Bölcskei*, Andrea Német-Hanzelik, Zsófia Dubrovay, Viktor Háda and György Keglevich
DOI: 10.2174/1570180816666181106123809

Synthesis, Antioxidant and Anti-inflammatory Activities of 5-((styrylsulfonyl) methyl)-1,3,4-Oxadiazol / Thiadiazol-2-amine Derivatives

Volume: 16   Issue: 11
Pp: 1233-1247
Gundala Sravya, Ummadi Nagarjuna, Venkatapuram Padmavathi, Galla Rajitha, Sakuri Chandi priya and Adivireddy Padmaja*
DOI: 10.2174/1570180816666181102114529

Design, Synthesis and Pharmacological Evaluation of Novel Antiinflammatory and Analgesic O-Benzyloxime Compounds Derived From Natural Eugenol

Volume: 16   Issue: 10
Pp: 1157-1166
Rodrigo César da Silva, Fabiano Veiga, Fabiana Cardoso Vilela, André Victor Pereira, Thayssa Tavares da Silva Cunha, Roberta Tesch, Claudio Viegas Jr., Danielle Ferreira Dias, Alexandre Giusti-Paiva, Marcia Paranho Veloso and Carlos Alberto Manssour Fraga*
DOI: 10.2174/1570180815666180620145609

Benzo[d]imidazol-5-yl)-5-(substituted)-1,3,4-Oxadiazoles: Synthesis, Anticancer, Antimicrobial and In Silico Studies open access plus

Volume: 16   Issue: 9
Pp: 994-1005
Naveen Kumar, Swamy Sreenivasa*, Bhuvanesh Sukhlal Kalal, Vasantha Kumar, Bantwal Shivarama Holla, Vinitha Ramanath Pai, Nadigar Revansiddappa Mohan and Shivaraj Govindaiah
DOI: 10.2174/1570180816666181220123924

Paclitaxel-tyroserleutide Conjugates Self-assembly into Nanocarrier for Drug Delivery

Volume: 16   Issue: 8
Pp: 882-891
Yongjia Liu, Leilei Shi, Bangshang Zhu*, Yue Su, Hui Li* and Xinyuan Zhu
DOI: 10.2174/1570180815666180803124625

Design, Synthesis, Biological Evaluation and In Silico Studies of Few Novel 2-Substituted Benzothiazole Derivatives as Potential EGFR Inhibitors

Volume: 16   Issue: 8
Pp: 961-971
Muhammad Mubeen, Suvarna Ganesh Kini*, Avinash Kumar and Karkala Sreedhara Ranganath Pai
DOI: 10.2174/1570180816666181108112228

Design, Synthesis and Biological Evaluation of Camptothecin Conjugated with NSAIDs as Novel Dual-actin Antitumor Agents

Volume: 16   Issue: 12
Pp: 1378-1386
Xingchen Cai, Weiwei Huang, Yi Huang, Lihua Xia, Miao Liu, Mengke Wang, Wenchao Wang and Qingyong Li*
DOI: 10.2174/1570180816666190221103257