Medicinal Chemistry

Editor-in-Chief:

Dimitra Hadjipavlou-Litina
Aristotle University of Thessaloniki
Thessaloniki
Greece

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Graphical Abstracts: promotion: free to download

Volume:9   Issue:8
Pp: i-v

DOI: 10.2174/1573406411309080001

Hemisynthesis of Selected Embelin Analogs and Investigation of their Proapoptotic Activity Against Cancer Cells

Volume:9   Issue:8
Pp: 1028-1034
Guillaume Viault, Katragadda Suresh Babu, Fabien Gautier, Sophie Barillé-Nion, Philippe Juin, Olivier Tasseau and René Grée
DOI: 10.2174/1573406411309080003

Synthesis and Inhibitory Effects of Some Novel 1,3-diarylprop-2-en-1-one Analogues in Foxp3 Expression: A Novel Class of Anti-cancer Candidates

Volume:9   Issue:8
Pp: 1035-1040
Mayank Kinger, Jeong Hoon Park, Min Goo Hur, Sang Wook Kim and Seung Dae Yang
DOI: 10.2174/15734064113099990029

New Benzothiazole/thiazole-Containing Hydroxamic Acids as Potent Histone Deacetylase Inhibitors and Antitumor Agents

Volume:9   Issue:8
Pp: 1051-1057
Truong Thanh Tung, Dao Thi Kim Oanh, Phan Thi Phuong Dung, Van Thi My Hue, Sang Ho Park, Byung Woo Han, Youngsoo Kim, Jin-Tae Hong, Sang-Bae Han and Nguyen-Hai Nam
DOI: 10.2174/15734064113099990027

Synthesis and Anti-tumor Activity Evaluation of Gallic Acid-mangiferin Hybrid Molecule

Volume:9   Issue:8
Pp: 1058-1062
Xiang-yu Hu, Jia-gang Deng, Lin Wang and Ye-fei Yuan
DOI: 10.2174/1573406411309080007

Synthesis and in vitro Cytotoxicity Studies of Certain Novel Heterocycles Derived from Bis 1, 2, 4-Triazoles and their DNA Damage Studies

Volume:9   Issue:8
Pp: 1063-1072
Madhusudan N. Purohit, Chandrashekhar Venkaraddi Mangannavar and Mayur C. Yergeri
DOI: 10.2174/1573406411309080008

QSAR and Docking Based Semi-synthesis and in vitro Evaluation of 18 β-glycyrrhetinic Acid Derivatives Against Human Lung Cancer Cell Line A-549

Volume:9   Issue:8
Pp: 1073-1084
Dharmendra Kumar Yadav, Komal Kalani, Feroz Khan and Santosh Kumar Srivastava
DOI: 10.2174/1573406411309080009

Synthesis of 1H-1,2,3-triazoles and Study of their Antifungal and Cytotoxicity Activities

Volume:9   Issue:8
Pp: 1085-1090
Iara F. da Silva, Prisicila R.C. Martins, Emanuelly G. da Silva, Sabrina B. Ferreira, Vitor F. Ferreira, Karen Regina C. da Costa, Marne C. de Vasconcellos, Emerson S. Lima and Fernando de C. da Silva
DOI: 10.2174/1573406411309080010

Synthesis and Effects of Pyrazolines and Isoxazoles on the Phagocytic Chemotaxis and Release of Reactive Oxygen Species by Zymosan Stimulated Human Neutrophils

Volume:9   Issue:8
Pp: 1091-1098
Syed Nasir Abbas Bukhari, Ibrahim Jantan, Lam Kok Wai, Nordin Haji Lajis, Faridah Abbas and Malina Jasamai
DOI: 10.2174/1573406411309080011

Synthesis and Biological Evaluation of Some Novel Thieno[2,3-d] pyrimidine Derivatives as Potential Anti-inflammatory and Analgesic Agents

Volume:9   Issue:8
Pp: 1099-1112
Alaa A. El-Tombary, Soad A.M. El-Hawash, Nargues S. Habib, Raafat Soliman, Ibrahim M. El-Ashmawy and Omaima G. Shaaban
DOI: 10.2174/1573406411309080012

Design, Synthesis, and Bioactivity of Pyrazole Acid Derivatives as Endothelin Receptor Antagonists

Volume:9   Issue:8
Pp: 1113-1122
Jin Cai, Ligang Liu, Junqing Chen, Meng Cao and Min Ji
DOI: 10.2174/1573406411309080013

Effect of Stabilizers on Bioactivity of Peptide-24 in PLGA Microspheres

Volume:9   Issue:8
Pp: 1123-1128
Mingbo Wang, XiaoDong Guo, Rongwei Tan, Zhending She and Qingling Feng
DOI: 10.2174/1573406411309080014

Synthesis and in vitro Antibacterial Activity of 5-Halogenomethylsulfonyl- Benzimidazole and Benzotriazole Derivatives

Volume:9   Issue:8
Pp: 1129-1136
Zbigniew Ochal, Maria Bretner, Renata Wolinowska and Stefan Tyski
DOI: 10.2174/1573406411309080015

ACKNOWLEDGEMENT TO REVIEWERS: promotion: free to download

Volume:9   Issue:8
Pp: 1137-1137

DOI: 10.2174/1573406411309080016