Medicinal Chemistry

Editor-in-Chief:

Dimitra Hadjipavlou-Litina
Aristotle University of Thessaloniki
Thessaloniki
Greece

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Volume:9   Issue: 7
Pp: i-vi

DOI: 10.2174/1573406411309070001

Current Prospects of Synthetic Curcumin Analogs and Chalcone Derivatives Against Mycobacterium Tuberculosis

Volume:9   Issue: 7
Pp: 897-903
Syed Nasir Abbas Bukhari, Scott G. Franzblau, Ibrahim Jantan and Malina Jasamai
DOI: 10.2174/1573406411309070002

Increment of Antimycobaterial Activity on Lichexanthone Derivatives

Volume:9   Issue: 7
Pp: 904-910
Ana Camila Micheletti, Neli Kika Honda, Fernando R. Pavan, Clarice Q. F. Leite, Maria de Fatima Cepa Matos, Renata Trentin Perdomo, Danielle Bogo, Glaucia Braz Alcantara and Adilson Beatriz
DOI: 10.2174/1573406411309070003

Aromatic Sulfonamides Containing a Condensed Piperidine Moiety as Potential Oxidative Stress-Inducing Anticancer Agents

Volume:9   Issue: 7
Pp: 911-919
Ramóna Madácsi, Iván Kanizsai, Liliána Z. Fehér, Márió Gyuris, Béla Ózsvári, András Erdélyi, János Wölfling and László G. Puskás
DOI: 10.2174/1573406411309070004

Synthesis and Biological Activity of 28-Amide Derivatives of 23-Hydroxy Betulinic Acid as Antitumor Agent Candidates

Volume:9   Issue: 7
Pp: 920-925
Yi Bi, Jinyi Xu, Fei Sun, Xiaoming Wu, Wencai Ye, Yijun Sun and Wenwen Huang
DOI: 10.2174/1573406411309070005

Dynamic Function of the Alkyl Spacer of Acetogenins as Potent Inhibitors of Mitochondrial Complex I. A Molecular Dynamics Simulation Approach

Volume:9   Issue: 7
Pp: 926-937
José Abel Bombasaro, Exequiel Ernesto Barrera Guisasola, Marcelo Fabricio Masman, Miguel Angel Zamora and Ana María Rodríguez
DOI: 10.2174/1573406411309070006

Design, Synthesis and Biological Evaluation of Novel Imidazolone Derivatives as Dipeptidyl Peptidase 4 Inhibitors

Volume:9   Issue: 7
Pp: 938-946
Yang Liu, Chaoyi Jiang, Haoshu Wu, Peng Wu, Meimei Si, Yongzhou Hu and Tao Liu
DOI: 10.2174/1573406411309070007

Design, Synthesis and Biological Evaluation of Ferulic Acid Amides as Selective Matrix Metalloproteinase Inhibitors

Volume:9   Issue: 7
Pp: 947-954
Zhi-Hao Shi, Nian-Guang Li, Qian-Ping Shi, Hao-Tang, Yu-Ping Tang, Wei-Li, Lian-Yin, Jian-Ping Yang and Jin-Ao Duan
DOI: 10.2174/1573406411309070008

Arylazolylthioacetanilide. Part 11: Design, Synthesis and Biological Evaluation of 1,2,4-triazole Thioacetanilide Derivatives as Novel Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors

Volume:9   Issue: 7
Pp: 968-973
Zhenyu Li, Yuan Cao, Peng Zhan, Christophe Pannecouque, Jan Balzarini, Erik De Clercq, Yuemao Shen and Xinyong Liu
DOI: 10.2174/1573406411309070010

Pharmacophore Based 3D-QSAR Study of Biphenyl Derivatives as Nonsteroidal Aromatase Inhibitors in JEG-3 Cell Lines

Volume:9   Issue: 7
Pp: 974-984
Lakshmi Narayana Bheemanapalli, Balakumar C, Venkat Rao Kaki, Rajwinder Kaur and Raghuram Rao Akkinepally
DOI: 10.2174/1573406411309070011

Molecular Simulation to Investigate the Cofactor Specificity for Pichia stipitis Xylose Reductase

Volume:9   Issue: 7
Pp: 985-992
Xiao-Le Xia, Shan Cong, Xiao-Rong Weng, Jin-Hua Chen, Jing-Fang Wang and Kuo-Chen Chou
DOI: 10.2174/1573406411309070012

Structural Modeling and Identification of Imperatorin as Novel L-type Calcium Channel Blocker

Volume:9   Issue: 7
Pp: 993-998
Wen Lu, Tao Zhang, Pengfei Li, Fang Wang, Xiaoyan Pan, Chen Wang, Zhigang Hu and Jie Zhang
DOI: 10.2174/1573406411309070013

Curcumin Bioconjugates: Studies on Structure-Activity Relationship and Antibacterial Properties against Clinically Isolated Strains

Volume:9   Issue: 7
Pp: 999-1005
Diwakar Rai, Garima Kumari, Anuradha Singh and Ramendra K. Singh
DOI: 10.2174/1573406411309070014

Synthesis and Evaluation of Antioxidant-S-(+)-Ibuprofen Hybrids as Gastro Sparing NSAIDs

Volume:9   Issue: 7
Pp: 1006-1016
Senthil Chandiran, Sandeep Vyas, Neetika Sharma and Manu Sharma
DOI: 10.2174/1573406411309070015