Medicinal Chemistry

Dimitra Hadjipavlou-Litina
Aristotle University of Thessaloniki
Thessaloniki
Greece

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Synthesis and Biological Evaluation of 3΄-C-Ethynyl and 3΄-C-(1,4-disubstituted-1,2,3-triazolo) Double-Headed Pyranonucleosides

Volume:8   Issue:3
Pp: 320-329
Christos Kiritsis, Stella Manta, Ioannis Papasotiriou, Evdoxia Coutouli-Argyropoulou, Sakellarios Trakossas, Jan Balzarini and Dimitri Komiotis
DOI: 10.2174/157340612800786624

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Substituted Urea Derivatives: A Potent Class of Antidepressant Agents

Volume:8   Issue:3
Pp: 330-336
Shahnaz Perveen, Sana Mustafa, Muhammad A. Khan, Ahsana Dar, Khalid M. Khan and Wolfgang Voelter
DOI: 10.2174/157340612800786615

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SAR Analysis of New Dual Targeting Fluoroquinolones. Implications of the Benzenesulfonyl Group

Volume:8   Issue:3
Pp: 349-360
Marcelo J. Nieto, Adriana B. Pierini, Nidhi Singh, Christopher R. McCurdy, Ruben H. Manzo and aria R. Mazzieri
DOI: 10.2174/157340612800786633

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S-Nitrosylation and Attenuation of Excessive Calcium Flux by Pentacycloundecane Derivatives

Volume:8   Issue:3
Pp: 361-371
Hendrik J.R. Lemmer, Jacques Joubert, Sandra van Dyk, Francois H. van der Westhuizen and Sarel F. Malan
DOI: 10.2174/1573406411208030361

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CoMFA and CoMSIA Studies of 1,2-dihydropyridine Derivatives as Anticancer Agents

Volume:8   Issue:3
Pp: 372-383
Ismail Salama, Mohamed A. O. Abdel-Fattah, Marwa S. Hany, Shaimaa A. El-Sharif, Mahmoud A. M. El-Naggar, Rasha M. H. Rashied, Gary A. Piazza and Ashraf H. Abadi
DOI: 10.2174/157340612800786598

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Four-Component Synthesis of 1,2-Dihydropyridine Derivatives and their Evaluation as Anticancer Agents

Volume:8   Issue:3
Pp: 392-400
Mohamed A. O. Abdel-Fattah, Mahmoud A. M. El-Naggar, Rasha M. H. Rashied, Bernard D. Gary, Gary A. Piazza and Ashraf H. Abadi
DOI: 10.2174/1573406411208030392

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Biological and Anti-inflammatory Evaluation of Two Thiazole Compounds in RAW Cell Line: Potential Cyclooxygenase-2 Specific Inhibitors

Volume:8   Issue:3
Pp: 401-408
Eva Hamade, Aida Habib, Ali Hachem, Alaa H. Hussein, Malak Abbas, Taghreed Hirz, Mirvat Al Masri and Wissam H. Faour
DOI: 10.2174/1573406411208030401

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In vitro Anti-glycation and Anti-oxidant Properties of Synthesized Schiff Bases

Volume:8   Issue:3
Pp: 409-414
Sabina Jhaumeer-Laulloo, Minu Gupta Bhowon, Shabneez Mungur, Mohamad Fawzi Mahomoodally and Anwar Hussein Subratty
DOI: 10.2174/1573406411208030409

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Synthesis and Antiglycation Activity of Kaempferol-3-O-rutinoside (Nicotiflorin)

Volume:8   Issue:3
Pp: 415-420
Sajan Lal Shyaula, Ghulam Abbas, Hina Siddiqui, Samina A. Sattar, M. Iqbal Choudhary and Fatima Z. Basha
DOI: 10.2174/1573406411208030415

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Synthesis and β-Glucuronidase Inhibitory Potential of Benzimidazole Derivatives

Volume:8   Issue:3
Pp: 421-427
Khalid Mohammed Khan, Momin Khan, Nida Ambreen, Fazal Rahim, Shagufta Naureen, Shahnaz Perveen, M. Iqbal Choudhary and Wolfgang Voelter
DOI: 10.2174/1573406411208030421

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Design, Synthesis and Evaluation of Unique 2,4,5-triaryl Imidazole Derivatives as Novel Potent Aspartic Protease Inhibitors

Volume:8   Issue:3
Pp: 428-435
Mohd Sajid Khan, Salman Akhtar, S. A. Siddiqui, M. S. Siddiqui, K. V. Srinivasan and J. M. Arif
DOI: 10.2174/1573406411208030428

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2,4,6-Trichlorophenylhydrazine Schiff Bases as DPPH Radical and Super Oxide Anion Scavengers

Volume:8   Issue:3
Pp: 452-461
Khalid Mohammed Khan, Zarbad Shah, Viqar Uddin Ahmad, Momin Khan, Muhammad Taha, Fazal Rahim, Sajjad Ali, Nida Ambreen, Shahnaz Perveen, M. Iqbal Choudhary and Wolfgang Voelter
DOI: 10.2174/1573406411208030452

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Structure-Activity Relationships of Pyrrole Hydrazones as New Anti-Tuberculosis Agents

Volume:8   Issue:3
Pp: 462-473
Iglika Lessigiarska, Ilza Pajeva, Penka Prodanova, Maya Georgieva and Atanas Bijev
DOI: 10.2174/1573406411208030462

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Synthesis and Biological Evaluation of the Salicylamide and Salicylic Acid Derivatives as Anti-Estrogen Agents

Volume:8   Issue:3
Pp: 481-490
Yasemin Dundar, Yasemin Ozatik, Orhan Ozatik, Volkan Ergin, Tijen Onkol, Adnan Menevse, Kevser Erol and M. Fethi Sahin
DOI: 10.2174/1573406411208030481

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Synthesis and Biological Evaluation of Some New N4-Aryl Substituted 5-Chloroisatin-3-thiosemicarbazones

Volume:8   Issue:3
Pp: 505-514
Humayun Pervez, Muhammad Ramzan, Muhammad Yaqub, Faiz-ul-Hassan Nasim and Khalid Mohammed Khan
DOI: 10.2174/1573406411208030505

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