Medicinal Chemistry

Editor-in-Chief:

Dimitra Hadjipavlou-Litina
Aristotle University of Thessaloniki
Thessaloniki
Greece

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Styrylquinoline – A Versatile Scaffold in Medicinal Chemistry

Volume:16   Issue: 2
Pp: 141-154
Robert Musiol*
DOI: 10.2174/1573406415666190603103012



Target Based Virtual Screening of New Leads Inhibitor against Bacterial Cell Division Protein FtsZ for the Discovery of Antibacterial Agents

Volume:16   Issue: 2
Pp: 169-175
Ratish C. Mishra, Rosy Kumari, Shivani Yadav and Jaya P. Yadav*
DOI: 10.2174/1573406415666190206233448



Design and Synthesis of New Substituted Pyrazolopyridines with Potent Antiproliferative Activity

Volume:16   Issue: 2
Pp: 176-191
Vassiliki Giannouli, Nikolaos Lougiakis, Ioannis K. Kostakis, Nicole Pouli*, Panagiotis Marakos, Alexios-Leandros Skaltsounis, David A. Horne, Sangkil Nam, Katerina Gioti and Roxane Tenta
DOI: 10.2174/1573406415666190222130225



Bicycloheptylamine-Doxorubicin Conjugate: Synthesis and Anticancer Activities in σ2 Receptor-Expressing Cell Lines

Volume:16   Issue: 2
Pp: 192-201
Mohammed A. Alamri, Zeynep Ates-Alagoz and Adeboye Adejare*
DOI: 10.2174/1573406415666190301145203



Design, Synthesis, and Evaluation of Isoquinoline Ureas as TRPV1 Antagonists

Volume:16   Issue: 2
Pp: 202-211
Nehaben A. Gujarati, Bradley J. Undem and Vijaya L. Korlipara*
DOI: 10.2174/1573406415666190626130453



Novel p-Functionalized Chromen-4-on-3-yl Chalcones Bearing Astonishing Boronic Acid Moiety as MDM2 Inhibitor: Synthesis, Cytotoxic Evaluation and Simulation Studies

Volume:16   Issue: 2
Pp: 212-228
Richa Kaur Bhatia*, Lakhwinder Singh, Ruchika Garg, Maninder Kaur, Manmohan Yadav, Jitender Madan, Satyavathi Kancherla, Raghuvir R. S. Pissurlenkar and Evans C. Coutinho
DOI: 10.2174/1573406415666190531123751



4-Aminocoumarin based Aroylthioureas as Potential Jack Bean Urease Inhibitors; Synthesis, Enzyme Inhibitory Kinetics and Docking Studies

Volume:16   Issue: 2
Pp: 229-243
Tanzeela A. Fattah, Aamer Saeed, Zaman Ashraf, Qamar Abbas, Pervaiz A. Channar, Fayaz A. Larik and Mubashir Hassan
DOI: 10.2174/1573406415666190715164834



Synthesis of β-Ketosulfone Derivatives As New Non-Cytotoxic Urease Inhibitors In Vitro

Volume:16   Issue: 2
Pp: 244-255
Sarosh Iqbal*, Ajmal Khan, Rashid Nazir, Shumaila Kiran, Shahnaz Perveen, Khalid Mohammed Khan* and M. Iqbal Choudhary*
DOI: 10.2174/1573406415666190415163309



Synthesis, Biological Evaluation and Molecular Dynamics Simulation Studies of Novel Diphenyl Ethers

Volume:16   Issue: 2
Pp: 256-270
Amol B. Khade, Sidhartha S. Kar, Cinu Thomas A, Ashutosh Tiwari, Mradul Tiwari, Vandana K. E., Pritesh Bhat, Varadaraj Bhat G. and G. Gautham Shenoy*
DOI: 10.2174/1573406415666190306152907