Medicinal Chemistry

Editor-in-Chief:

Dimitra Hadjipavlou-Litina
Aristotle University of Thessaloniki
Thessaloniki
Greece

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Volume:15   Issue: 4
Pp: 327-327
Andreas Hilgeroth
DOI: 10.2174/157340641504190403151530



Rational Design of Colchicine Derivatives as anti-HIV Agents via QSAR and Molecular Docking

Volume:15   Issue: 4
Pp: 328-340
Apilak Worachartcheewan*, Napat Songtawee, Suphakit Siriwong, Supaluk Prachayasittikul*, Chanin Nantasenamat and Virapong Prachayasittikul
DOI: 10.2174/1573406414666180924163756



Phenolic Imidazole Derivatives with Dual Antioxidant/Antifungal Activity: Synthesis and Structure-Activity Relationship

Volume:15   Issue: 4
Pp: 341-351
Ana P. Bettencourt, Marián Castro, João P. Silva, Francisco Fernandes, Olga P. Coutinho, Maria J. Sousa, Maria Fernanda Proença* and Filipe M. Areias*
DOI: 10.2174/1573406414666181005143431



New N,C-Diaryl-1,2,4-triazol-3-ones: Synthesis and Evaluation as Anticancer Agents

Volume:15   Issue: 4
Pp: 360-372
Dolores Santa María*, Rosa M. Claramunt, José Elguero, Miguel Carda*, Eva Falomir and Celia Martín-Beltrán
DOI: 10.2174/1573406414666180821103604



Spirocyclohexadienones as an Uncommon Scaffold for Acetylcholinesterase Inhibitory Activity

Volume:15   Issue: 4
Pp: 373-382
Ralph C. Gomes, Renata P. Sakata*, Wanda P. Almeida* and Fernando Coelho*
DOI: 10.2174/1573406414666181109114214



Design, Synthesis and Anxiolytic Activity Evaluation of N-Acyltryptophanyl- Containing Dipeptides, Potential TSPO Ligands#

Volume:15   Issue: 4
Pp: 383-399
Tatiana A. Gudasheva*, Olga A. Deeva, Grigory V. Mokrov, Alina S. Dyabina, Milada A. Yarkova and Sergey B. Seredenin
DOI: 10.2174/1573406415666181119164846



Synthesis and Evaluation of Antifungal and Antitrypanosomastid Activities of Symmetrical 1,4-Disubstituted-1,2,3-Bistriazoles Obtained by CuAAC Conditions

Volume:15   Issue: 4
Pp: 400-408
Mauricio M. Victor*, Ravir R. Farias, Danielle L. da Silva, Paulo H.F. do Carmo, Maria A. de Resende-Stoianoff, Cláudio Viegas, Patrícia F. Espuri and Marcos J. Marques
DOI: 10.2174/1573406414666181024111522



Antiprotozoal Activities of Tetrazole-quinolines with Aminopiperidine Linker

Volume:15   Issue: 4
Pp: 409-416
Patrick Hochegger, Johanna Faist, Werner Seebacher, Robert Saf, Pascal Mäser, Marcel Kaiser and Robert Weis*
DOI: 10.2174/1573406414666181015115101



Ligand-Based Drug Design: Synthesis and Biological Evaluation of Substituted Benzoin Derivatives as Potential Antitumor Agents

Volume:15   Issue: 4
Pp: 417-429
Dima A. Sabbah*, Ameerah H. Ibrahim, Wamidh H. Talib, Khalid M. Alqaisi, Kamal Sweidan, Sanaa K. Bardaweel, Ghassan A. Sheikha, Haizhen A. Zhong, Eveen Al-Shalabi, Reema A. Khalaf and Mohammad S. Mubarak
DOI: 10.2174/1573406414666180912111846



Novel Conjugated Unsaturated Ketones with Submicromolar Potencies Towards some Leukemic and Colon Cancer Cells

Volume:15   Issue: 4
Pp: 430-438
Swagatika Das, H. Inci Gul, Umashankar Das*, Jan Balzarini, Stephen G. Dimmock and Jonathan R. Dimmock *
DOI: 10.2174/1573406414666181015142633