Medicinal Chemistry

Editor-in-Chief:

Dimitra Hadjipavlou-Litina
Aristotle University of Thessaloniki
Thessaloniki
Greece

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Volume:15   Issue: 1
Pp: 1-1
Dimitra Hadjipavlou-Litina
DOI: 10.2174/157340641501181122103125



Meet Our Editor-in-Chief free to download

Volume:15   Issue: 1
Pp: 2-2
Dimitra Hadjipavlou-Litina
DOI: 10.2174/157340641501181122103339



Sorbinil, an Aldose Reductase Inhibitor, in Fighting Against Diabetic Complications

Volume:15   Issue: 1
Pp: 3-7
Qi Huang, Qiong Liu and Dongsheng Ouyang*
DOI: 10.2174/1573406414666180524082445



Pyrano[3,2-c]quinoline Derivatives as New Class of α-glucosidase Inhibitors to Treat Type 2 Diabetes: Synthesis, in vitro Biological Evaluation and Kinetic Study

Volume:15   Issue: 1
Pp: 8-16
Zahra Heydari, Maryam Mohammadi-Khanaposhtani, Somaye Imanparast, Mohammad A. Faramarzi, Mohammad Mahdavi *, Parviz R. Ranjbar* and Bagher Larijani
DOI: 10.2174/1573406414666180528110104



Pyrazole and imidazo[1,2-b]pyrazole Derivatives as New Potential Antituberculosis Agents

Volume:15   Issue: 1
Pp: 17-27
Elda Meta, Chiara Brullo*, Michele Tonelli, Scott G. Franzblau, Yuehong Wang, Rui Ma, Wan Baojie, Beatrice S. Orena, Maria R. Pasca and Olga Bruno
DOI: 10.2174/1573406414666180524084023



4-Hydroxy-2-pyridone Derivatives and the δ-pyrone Isostere as Novel Agents Against Mycobacterium smegmatis Biofilm Inhibitors

Volume:15   Issue: 1
Pp: 28-37
Maheshkumar R. Borkar, Santosh Nandan*, Harish K.M. Nagaraj, Jayashree Puttur, Jisha Manniyodath, Dipankar Chatterji and Evans C. Coutinho *
DOI: 10.2174/1573406414666180525075755



Synthesis and Evaluation of the in vitro Antimicrobial Activity of Triazoles, Morpholines and Thiosemicarbazones

Volume:15   Issue: 1
Pp: 38-50
Felipe R.S. Santos, Jéssica T. Andrade, Carla D.F. Sousa, Joice S. Fernandes, Lucas F. Carmo, Marcelo G.F. Araújo, Jaqueline M.S. Ferreira and José A.F.P. Villar*
DOI: 10.2174/1573406414666180730111954



The Evaluation of Metal Co-ordinating Bis-Thiosemicarbazones as Potential Anti-malarial Agents

Volume:15   Issue: 1
Pp: 51-58
Fady N. Akladios, Scott D. Andrew, Samantha J. Boog, Carmen de Kock, Richard K. Haynes and Christopher J. Parkinson*
DOI: 10.2174/1573406414666180525132204



Design, Synthesis and Investigation of New Diphenyl Substituted Pyridazinone Derivatives as Both Cholinesterase and Aβ-Aggregation Inhibitors

Volume:15   Issue: 1
Pp: 59-76
Burcu Kilic, Merve Erdogan, Hayrettin O. Gulcan, Fatma Aksakal, Nihan Oruklu, Emin U. Bagriacik and Deniz S. Dogruer*
DOI: 10.2174/1573406414666180524073241



Synthesis and Biological Evaluation of Novel 2,3-disubstituted Benzofuran Analogues of GABA as Neurotropic Agents

Volume:15   Issue: 1
Pp: 77-86
Arturo Coaviche-Yoval, Héctor Luna, Ricardo Tovar-Miranda, Marvin A. Soriano-Ursúa and José G. Trujillo-Ferrara*
DOI: 10.2174/1573406414666180524091745



New Hybrid Scaffolds based on Hydrazinyl Thiazole Substituted Coumarin; As Novel Leads of Dual Potential; In Vitro α-Amylase Inhibitory and Antioxidant (DPPH and ABTS Radical Scavenging) Activities

Volume:15   Issue: 1
Pp: 87-101
Uzma Salar, Khalid M. Khan*, Sridevi Chigurupati, Shazia Syed, Shantini Vijayabalan, Abdul Wadood, Muhammad Riaz, Mehreen Ghufran and Shahnaz Perveen
DOI: 10.2174/1573406414666180903162243



Neuropharmacological Screening of Chiral and Non-chiral Phthalimide- Containing Compounds in Mice: in vivo and in silico Experiments

Volume:15   Issue: 1
Pp: 102-118
Carolina Campos-Rodríguez, José G. Trujillo-Ferrara*, Ameyali Alvarez-Guerra, Irán M. Cumbres Vargas, Roberto I. Cuevas-Hernández, Erik Andrade-Jorge, Sergio Zamudio and Eduardo R.-S. Juan*
DOI: 10.2174/1573406414666180525082038