Anti-Cancer Agents in Medicinal Chemistry

(Formerly Current Medicinal Chemistry - Anti-Cancer Agents)

This journal supports open access

Editor-in-Chief:

Michelle Prudhomme
Institut de Chimie de Clermont-Ferrand
ICCF-CNRS UMR 6296
Université Clermont Auvergne
Clermont-Ferrand
France

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Abstract Ahead of Print

Cytotoxic and genotoxic activities of alkaloids from the bulbs of Griffinia gardneriana and Habranthus itaobinus (Amaryllidaceae)

Volume:19
Eduardo R. Cole, Jean P. de Andrade, Joâo F. Allochio Filho, Elisângela F. P. Schmitt, Anderson Alves-Araújo, Jaume Bastida, Denise C. Endringer, Warley de S. Borges and Valdemar Lacerda*

Anti-Diarrheal Drug Repositioning in Tumour Cell Cytotoxicity

Volume:19
Jihene Elloumi-Mseddi, Dhouha Msalbi, Raouia Fakhfakh and Sami Aifa*

Adenosine analogues as opposite modulators of the cisplatin resistance of ovarian cancer cells

Volume:19
Katarzyna Bednarska-Szczepaniak*, Damian Krzyżanowski, Magdalena Klink* and Marek Nowak

Novel Fluorine Boron Hybrid Complex as Potential Antiproliferative Drugs on Colorectal Cancer Cell Line

Volume:19
Yasin Tülüce*, Hawro Dlawar Ismael Masseh, İsmail Koyuncu, Ahmet Kiliç, Mustafa Durgun and Halil Özkol

Tetrahydrocurcumin, Curcumin, and 5-Fluorouracil Effects on Human Esophageal Carcinoma Cells.

Volume:19
Emily Grace Pendleton, Roudabeh Jahromi Jamasbi and Michael Eric Geusz*

Synthesis and Screening of Pro-apoptotic and Angio-inhibitory Activity of Novel Benzisoxazole Derivatives Both In vitro and In vivo.

Volume:19
Sathish Byrappa, Kavitha Rachaiah, Sumana Y. Kotian, Yashaswini Balaraju, Samudyata C. Prabhuswamimath, K. M. Lokanatha Rai and Bharathi P. Salimath*

Nicotinamide Overcomes Doxorubicin Resistance of Breast Cancer Cells through Deregulating SIRT1/Akt Pathway

Volume:19
Yingze Wei, Yan Guo, Jianyun Zhou, Kui Dai, Qiang Xu and Xiaoxia Jin*

Isolation of a New Sesquiterpene Lactone From Vernonia Zeylanica (L) Less and its Anti-Proliferative Effects in Breast Cancer Cell Lines.

Volume:19
Anuka S Mendis*, M. Ira Thabrew, Meran K. Ediriweera, Sameera R Samarakoon, Kamani H Tennekoon, Achyut Adhikari* and E. Dilip de Silva

Design, Synthesis and Antiproliferative Evaluation of Novel 1,2,4-Triazole/Schiff Base Hybrids with EGFR and B-RAF Inhibitory Activities

Volume:19
Hany A. M. El-Sherief, Bahaa G. M. Youssif*, Ahmed H. Abdelazeem, Mohamed Abdel-Aziz and Hamdy M. Abdel-Rahman*

Influence of Resveratrol on Sphingolipid Metabolism in Hepatocellular Carcinoma Cells in Lipid Overload State

Volume:19
Tomasz Charytoniuk*, Ewa Harasim-Symbor , Agnieszka Polak, Krzysztof Drygalski, Klaudia Berk, Adrian Chabowski and Karolina Konstantynowicz-Nowicka

Let-7a could serve as a biomarker for chemoresistance against docetaxel in gastric cancer.

Volume:19
Tohid Kazemi*, Najibeh Shekari, Faezeh Asghari, Navideh Haghnavaz, Dariush Shanehbandi, Vahid Khaze and Behzad Baradaran

Berberine Effects on NFκB, HIF1A and NFE2L2/AP-1 Pathways in HeLa Cells

Volume:19
Anna Belanova , Darya Beseda , Victor Chmykhalo , Alisa Stepanova , Mariya Belousova , Vera Khrenkova , Nikolaos Gavalas and Peter Zolotukhin*

A Novel Camptothecin Derivative 3j Inhibits Nsclc Proliferation Via Induction of Cell Cycle Arrest By Topo I-Mediated DNA Damage

Volume:19
Yang Liu, Jingyin Zhang, Shuyun Feng, Tingli Zhao, Zhengzheng Li, Lai Wang, Puhai Wang, Hongzhi Du*, Shengtao Yuan* and Li Sun*

Novel Inhibitors of DNA Repair Enzyme TDP1 Combining Monoterpenoid and Adamantane Fragments.

Volume:19
Evgenii S. Mozhaitsev, Alexandra L. Zakharenko, Evgeniy V. Suslov*, Dina V. Korchagina, Olga D. Zakharova, Inna A. Vasil’eva, Arina A. Chepanova, Ellena Black, Jinal Patel, Raina Chand, Jóhannes Reynisson, Ivanhoe K. H. Leung, Konstantin P. Volcho, Nariman F. Salakhutdinov and Olga I. Lavrik

Induction of Apoptosis by pierisin-6 in HPV positive HeLa and HepG2 Cancer Cells is mediated by the caspase-3 dependent mitochondrial pathway.

Volume:19
Subbarayan Sarathbabu, Satheesh Kumar Marimuthu, Souvik Ghatak, Subramanian Vidyalakshmi, Gurusubramanian Guruswami, Sankar Kumar Ghosh, Selvi Subramanian, Wenqing Zhang and Nachimuthu Senthil Kumar*

Synthesis of 3-Arylaminopropenone Linked 2-Arylbenzo[d]imidazo[2,1-b]thiazole Conjugates as Anticancer and Apoptotic Inducing Agents

Volume:19
Ahmed Kamal*, Siddiq Pasha Shaik, T. Srinivasa Reddy, Satish Sunkari, A. V. Subba Rao and Korrapati Suresh Babu

Novel benzo[b]furans with anti-microtubule activity upregulate expression of apoptotic genes and arrest leukemia cells in G2/M phase

Volume:19
Karolina Kró lewska-Goliñska, Marcin J. Cieślak*, Milena Sobczak, Rafał Dolot, Ewa Radzikowska-Cieciura, Mariola Napiórkowska, Iwona Wybrañska and Barbara Nawrot

Single-chain antibody against Reg4 suppresses gastric cancer cell growth and enhances 5-FU-induced cell death in vitro

Volume:19
Xue-Qing Zhang , Lu-Ting Yu, Pei Du, Tian-Qi Yin, Zhi-Yuan Zhang, Ying Xu , Xiang Li, You-Jie Li , Min Wang* and Chen Luo *

Synthesis and In Vitro Evaluation of Tetrahydroquinoline Derivatives as Antiproliferative Compounds of Breast Cancer via Targeting The GPER

Volume:18
Oscar Jovan Zacarías-Lara, David Méndez-Luna, Gustavo Martínez-Ruíz, José Ruben García-Sanchéz, Manuel Jonathan Fragoso-Vázquez*, Martiniano Bello, Elvia Becerra-Martínez, Juan Benjamín García-Vázquez* and José Correa-Basurto*

Virtual screening of natural products to select compounds with potential anticancer activity

Volume:18
Élida Batista Vieira Sousa Cavalcanti, Mayara Barbalho FÉlix, Luciana Scotti* and Marcus Tullius Scottia

Integrins as A New Target for Cancer Treatment

Volume:18
Izabela Łasiñska* and Jacek Mackiewicz

Design, Synthesis and Evaluation of Novel 3/4-((Substituted benzamidophenoxy)methyl)-N-hydroxybenzamides / propenamides as Histone Deacetylase Inhibitors and Antitumor Agents

Volume:18
Duong Tien Anh, Nguyen Thi Thuan, Pham-The Hai, Le-Thi-Thu Huong, Nguyen Thi Kim Yen, Byung Woo Han, Eun Jae Park, Yeo Jin Choi, Jong Soon Kang, Van Thi My Hue*, Sang-Bae Han* and Nguyen-Hai Nam*

Hybridized quinoline derivatives as anticancer agents: Design, Synthesis, biological evaluation and molecular docking

Volume:18
Mohamed R. Selim, Medhat A. Zahran, Amany Belal*, Mostafa S. Mostafa*, Said A. Shedid, Ahmed B. M. Mehany, Gameel A. M. Elhagali and Yousry A. Ammar*

3, 3′-Dimethylquercetin Inhibits the Proliferation of Human Colon Cancer RKO Cells through Inducing G2/M Cell Cycle Arrest and Apoptosis

Volume:18
Jianguo Wu, Jun Yi, Yanbin Wu, Xuzheng Chen, Jianwei Zeng, Jinzhong Wu* and Wei Peng*

Cyclosporine A Suppresses the Malignant Progression of Oral Squamous Cell Carcinoma in vitro

Volume:18
Ling Gao, Jianwei Dong, Nanyang Zhang, Zhanxian Le, Wenhao Ren, Shaoming Li, Fan Li, Jianzhong Song, Qibo Wang, Zhichao Dou, Soo Young Park and Keqian Zhi*

Immunohistochemical expression of melatonin receptor MT1 and glucose transporter GLUT1 in human breast cancer

Volume:18
Tialfi Bergamin de Castro, André de Lima Mota, Newton Antônio Bordin-Junior, Dalisio de Santi Neto and Debora Aparecida Pires de Campos Zuccari*