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Letters in Drug Design & Discovery

Editor-in-Chief

ISSN (Print): 1570-1808
ISSN (Online): 1875-628X

Amide Mono Thioxylated Derivatives of MEN 10627

Author(s): M. Altamura, G. Balacco, A. Giolitti, A. Guidi, R. Patacchini, A. R. Renzetti, A. Triolo and C. A. Maggi

Volume 1 , Issue 3 , 2004

Page: [285 - 288] Pages: 4

DOI: 10.2174/1570180043398966

Price: $65

Abstract

The thioxylation of the potent Neurokinin A antagonist MEN 10627 by Lawessons reagent showed to be potentially useful for the post-synthetic manipulation of the related family of structurally peculiar bicyclic hexapeptides, whose synthesis in combinatorial manner has been recently described.

Keywords: tachykinins, thiopeptides, thioxopeptides, lawesson reagent, atp, anti-ischaemic drugs


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