Abstract
A new series of 1,2,4-triazoles containing cyclopropane moiety were synthesized and characterized by 1H NMR and elemental analyses. The biological activities results showed that most of them exhibited significant fungicidal activity towards six test fungi. Among them, several showed superiority over the commercial fungicide during the present study.
Keywords: 1, 2, 4-triazole, Cyclopropane, Antifungal activity, Synthesis, Microwave irradiation, Ultrasonic irradiation
Letters in Drug Design & Discovery
Title:Synthesis and Antifungal Activity of 1,2,4-triazole Derivatives Containing Cyclopropane Moiety
Volume: 9 Issue: 4
Author(s): Cheng-Xia Tan, Yan-Xia Shi, Jian-Quan Weng, Xing-Hai Liu, Bao-Ju Li, Wei-Guang Zhao
Affiliation:
Keywords: 1, 2, 4-triazole, Cyclopropane, Antifungal activity, Synthesis, Microwave irradiation, Ultrasonic irradiation
Abstract: A new series of 1,2,4-triazoles containing cyclopropane moiety were synthesized and characterized by 1H NMR and elemental analyses. The biological activities results showed that most of them exhibited significant fungicidal activity towards six test fungi. Among them, several showed superiority over the commercial fungicide during the present study.
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Cite this article as:
Cheng-Xia Tan, Yan-Xia Shi, Jian-Quan Weng, Xing-Hai Liu, Bao-Ju Li, Wei-Guang Zhao , Synthesis and Antifungal Activity of 1,2,4-triazole Derivatives Containing Cyclopropane Moiety, Letters in Drug Design & Discovery 2012; 9 (4) . https://dx.doi.org/10.2174/157018012799859954
DOI https://dx.doi.org/10.2174/157018012799859954 |
Print ISSN 1570-1808 |
Publisher Name Bentham Science Publisher |
Online ISSN 1875-628X |
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