New DNA Intercalating Acridinic Ligands: Comparative Copper-Catalyzed N-Arylation Reactions of 4-Aminoacridine with Organobismuth, Organoboron and Organolead Compounds

Author(s): Kamal Shimi, Gerard Boyer, Jean-Pierre Finet, Jean-Pierre Galy.

Journal Name: Letters in Organic Chemistry

Volume 1 , Issue 1 , 2004

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Abstract:

Copper diacetate catalyzed phenylation of 4-aminoacridine afforded the N-phenyl derivative in good yields with triphenylbismuth diacetate, moderate yields with phenylboronic acid and failed with in situ generated phenyllead triacetate. All systems gave high yields of the N-monophenyl derivative in their reaction with 3,4-dimethylaniline.

Keywords: aminoacridine, copper catalysis, organobismuth, organoboron, organolead

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Article Details

VOLUME: 1
ISSUE: 1
Year: 2004
Page: [34 - 36]
Pages: 3
DOI: 10.2174/1570178043488798

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