Catalysis and the Synthesis of Pharmacologically Small Molecules

Author(s): Mohammad A. Alam.

Journal Name: Current Organic Chemistry

Volume 23 , Issue 9 , 2019

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Zakeyah, A.A.; Whitt, J.; Duke, C.; Gilmore, D.F.; Meeker, D.G.; Smeltzer, M.S.; Alam, M.A. Synthesis and antimicrobial studies of hydrazone derivatives of 4-[3-(2,4-difluorophenyl)-4-formyl-1H-pyrazol-1-yl]benzoic acid and 4-[3-(3,4-difluorophenyl)-4-formyl-1H-pyrazol-1-yl]benzoic acid. Bioorg. Med. Chem. Lett., 2018, 28, 2914-2919.
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Whitt, J.; Duke, C.; Sumlin, A.; Chambers, S.A.; Alnufaie, R.; Gilmore, D.; Fite, T.; Basnakian, A.G.; Alam, M.A. Synthesis of Hydrazone Derivatives of 4-[4-Formyl-3-(2-oxochromen-3-yl)pyrazol-1-yl]benzoic acid as Potent Growth Inhibitors of Antibiotic-resistant Staphylococcus aureus and Acinetobacter baumannii. Molecules, 2019, 24, 2051.
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Ali, M.A.; Okolo, C.; Alsharif, Z.A.; Whitt, J.; Chambers, S.A.; Varma, R.S.; Alam, M.A. Benign Synthesis of Thiazolo-androstenone Derivatives as Potent Anticancer Agents. Org. Lett., 2018, 20, 5927-5932.
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Gurrapu, S.; Jonnalagadda, S.K.; Alam, M.A.; Ronayne, C.T.; Nelson, G.L.; Solano, L.N.; Lueth, E.A.; Drewes, L.R.; Mereddy, V.R. Coumarin carboxylic acids as monocarboxylate transporter 1 inhibitors: In vitro and in vivo studies as potential anticancer agents. Bioorg. Med. Chem. Lett., 2016, 26, 3282-3286.
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Alsharif, Z.A.; Alam, M.A. Modular synthesis of thiazoline and thiazole derivatives by using a cascade protocol. RSC Advances, 2017, 7, 32647-32651.
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Alam, M.A.; Alsharif, Z.; Alkhattabi, H.; Jones, D.; Delancey, E.; Gottsponer, A.; Yang, T. Hexafluoroisopropyl alcohol mediated synthesis of 2,3-dihydro-4H-pyrido[1,2-a]pyrimidin-4-ones. Sci. Rep., 2016, 6, 36316.
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Alsharif, Z.; Ali, M.A.; Alkhattabi, H.; Jones, D.; Delancey, E.; Ravikumar, P.C.; Alam, M.A. Hexafluoroisopropanol mediated benign synthesis of 2H-pyrido[1,2-a]pyrimidin-2-ones by using a domino protocol. New J. Chem., 2017, 41, 14862-14870.
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Tokeer, A.; Ruby, P.; Huma, K. Iron Oxide Nanoparticles: An Efficient Nano-catalyst. Curr. Org. Chem., 2019, 23, 992-1002.


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Article Details

VOLUME: 23
ISSUE: 9
Year: 2019
Page: [976 - 977]
Pages: 2
DOI: 10.2174/138527282309190710102427

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