Benzazepine, a seven membered aza-heterocyclic ring fused with aromatic unit, is involved
in research aimed to evaluate new products that possess interesting biological activities. The aim of
this review is to provide an overview of the diverse and important pharmacological activities of benzazepine
moiety. This review highlights importance of benzazepine derivatives as anti-depressant,
anti-hypertensive, anti-ischaemic, anorectic, anti-histamine agents, AChE inhibitor, TRPV1 antagonist
and also in the treatment of hyponatremia. Recent efforts made to discover various pharmacologically
active molecules that contain benzazepine moiety are also reported.